Activity-based protein profiling reveals off-target proteins of the FAAH inhibitor BIA 10-2474. (Q48304342)

http://europepmc.org/abstract/PMC/5641481

9 July 2018

title

Activity-based protein profiling reveals off-target proteins of the FAAH inhibitor BIA 10-2474. (English)

1 reference

http://europepmc.org/abstract/PMC/5641481

9 July 2018

author

Marc P Baggelaar

8

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:28596366%20AND%20SRC:MED&resulttype=core&format=json

31 May 2020

Thomas Hankemeier

23

1 reference

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31 May 2020

Annelot C M van Esbroeck

1

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31 May 2020

Antonius P A Janssen

2

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31 May 2020

Armand B Cognetta

3

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31 May 2020

Daisuke Ogasawara

4

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31 May 2020

Guy Shpak

5

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31 May 2020

Mark van der Kroeg

6

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31 May 2020

Vasudev Kantae

7

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31 May 2020

Femke M de Vrij

9

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31 May 2020

Hui Deng

10

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31 May 2020

Marco Allarà

11

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31 May 2020

Filomena Fezza

12

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31 May 2020

Zhanmin Lin

13

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31 May 2020

Tom van der Wel

14

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31 May 2020

Marjolein Soethoudt

15

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31 May 2020

Elliot D Mock

16

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31 May 2020

Hans den Dulk

17

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31 May 2020

Ilse L Baak

18

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31 May 2020

Bogdan I Florea

19

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31 May 2020

Giel Hendriks

20

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31 May 2020

Luciano De Petrocellis

21

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31 May 2020

Herman S Overkleeft

22

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31 May 2020

Vincenzo Di Marzo

25

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31 May 2020

Mauro Maccarrone

26

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31 May 2020

Benjamin Cravatt

27

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31 May 2020

Steven A Kushner

28

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31 May 2020

Mario van der Stelt

29

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31 May 2020

24

Chris I De Zeeuw

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31 May 2020

language of work or name

English

0 references

publication date

1 June 2017

1 reference

http://europepmc.org/abstract/PMC/5641481

9 July 2018

published in

Science

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31 May 2020

volume

356

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31 May 2020

issue

6342

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31 May 2020

page(s)

1084-1087

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:28596366%20AND%20SRC:MED&resulttype=core&format=json

Acute Neurologic Disorder from an Inhibitor of Fatty Acid Amide Hydrolase

31 May 2020

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Implications of the BIA-102474-101 study for review of first-into-human clinical trials

10 July 2018

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Rapid and profound rewiring of brain lipid signaling networks by acute diacylglycerol lipase inhibition

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Loss-of-function mutations in PNPLA6 encoding neuropathy target esterase underlie pubertal failure and neurological deficits in Gordon Holmes syndrome

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10 July 2018

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Discovery of PF-04457845: A Highly Potent, Orally Bioavailable, and Selective Urea FAAH Inhibitor

10 July 2018

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10 July 2018

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Superfamily-wide portrait of serine hydrolase inhibition achieved by library-versus-library screening

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10 July 2018

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10 July 2018

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14 August 2018

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14 August 2018

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14 August 2018

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14 August 2018

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Identifiers

DOI

10.1126/SCIENCE.AAF7497

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:28596366%20AND%20SRC:MED&resulttype=core&format=json

31 May 2020

1 reference

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31 May 2020

PubMed publication ID

28596366

1 reference