mGluR2 positive allosteric modulators: a patent review (2009 - present). (Q38085707)

28 August 2017

title

mGluR2 positive allosteric modulators: a patent review (2009 - present). (English)

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28 August 2017

Andrés A Trabanco

1

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author name string

José María Cid

series ordinal

2

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28 August 2017

language of work or name

English

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publication date

2 March 2013

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Expert Opinion on Therapeutic Patents

28 August 2017

published in

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28 August 2017

volume

23

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28 August 2017

issue

5

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28 August 2017

page(s)

629-647

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Metabotropic glutamate receptors: physiology, pharmacology, and disease

28 August 2017

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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Design and synthesis of an orally active metabotropic glutamate receptor subtype-2 (mGluR2) positive allosteric modulator (PAM) that decreases cocaine self-administration in rats

21 January 2018

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Orally active metabotropic glutamate subtype 2 receptor positive allosteric modulators: structure-activity relationships and assessment in a rat model of nicotine dependence

21 January 2018

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The mGlu2 but not the mGlu3 receptor mediates the actions of the mGluR2/3 agonist, LY379268, in mouse models predictive of antipsychotic activity

21 January 2018

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Use of MGLUR2 and MGLUR3 knockout mice to explore in vivo receptor specificity of the MGLUR2/3 selective antagonist LY341495.

21 January 2018

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Evidence for the role of metabotropic glutamate (mGlu)2 not mGlu3 receptors in the preclinical antipsychotic pharmacology of the mGlu2/3 receptor agonist (-)-(1R,4S,5S,6S)-4-amino-2-sulfonylbicyclo[3.1.0]hexane-4,6-dicarboxylic acid (LY404039).

21 January 2018

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10.1517/13543776.2013.777043

21 January 2018

Identifiers

DOI

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28 August 2017

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