GABAB receptor agonism as a novel therapeutic modality in the treatment of gastroesophageal reflux disease (Q37775213)

23 August 2017

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title

GABAB receptor agonism as a novel therapeutic modality in the treatment of gastroesophageal reflux disease (English)

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gastroesophageal reflux disease

23 August 2017

main subject

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author name string

Anders Lehmann

series ordinal

1

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23 August 2017

Jörgen M Jensen

series ordinal

2

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23 August 2017

Guy E Boeckxstaens

series ordinal

3

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23 August 2017

publication date

1 January 2010

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23 August 2017

published in

Advances in Pharmacology

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23 August 2017

volume

58

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23 August 2017

page(s)

287-313

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Synthesis and pharmacological evaluation of novel gamma-aminobutyric acid type B (GABAB) receptor agonists as gastroesophageal reflux inhibitors

23 August 2017

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3-Aminopropylphosphinic acid--a potent, selective GABAB receptor agonist in the guinea-pig ileum and rat anococcygeus muscle

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7 January 2021

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7 January 2021

Activation of the GABA(B) receptor inhibits transient lower esophageal sphincter relaxations in dogs

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7 January 2021

(R)-(3-amino-2-fluoropropyl) phosphinic acid (AZD3355), a novel GABAB receptor agonist, inhibits transient lower esophageal sphincter relaxation through a peripheral mode of action

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Characteristics and Frequency of Transient Relaxations of the Lower Esophageal Sphincter in Patients With Reflux Esophagitis

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Triggering of transient LES relaxations in ferrets: role of sympathetic pathways and effects of baclofen

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G-Protein-coupled modulation of presynaptic calcium currents and transmitter release by a GABAB receptor

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The Montreal definition and classification of gastroesophageal reflux disease: a global evidence-based consensus

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Excess gastroesophageal reflux in patients with hiatus hernia is caused by mechanisms other than transient LES relaxations

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Heterodimerization is required for the formation of a functional GABA(B) receptor

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Review of the quality of life and burden of illness in gastroesophageal reflux disease

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Gastroesophageal reflux symptoms and well-being in a random sample of the general population of a Swedish community

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7 January 2021

Functional GABAB receptors are present in guinea pig nodose ganglion cell bodies but not in peripheral mechanosensitive endings.

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7 January 2021

Control of transient lower oesophageal sphincter relaxations and reflux by the GABA(B) agonist baclofen in patients with gastro-oesophageal reflux disease

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7 January 2021

10.1016/S1054-3589(10)58012-8

Identifiers

DOI

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23 August 2017

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