Synthesis of novel antimitotic agents based on 2-amino-3-aroyl-5-(hetero)arylethynyl thiophene derivatives (Q35008501)

5 August 2017

title

Synthesis of novel antimitotic agents based on 2-amino-3-aroyl-5-(hetero)arylethynyl thiophene derivatives (English)

1 reference

5 August 2017

Stefania Grimaudo

7

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Andrea Brancale

Andrea Brancale

9

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Rosaria Maria Pipitone

Rosaria Maria Pipitone

6

0 references

Jan Balzarini

8

Jan Balzarini

1 reference

5 August 2017

Antonietta Di Cristina

5

Antonietta Di Cristina

1 reference

5 August 2017

4

Manlio Tolomeo

1 reference

5 August 2017

Romeo Romagnoli

1

1 reference

5 August 2017

Pier Giovanni Baraldi

2

1 reference

5 August 2017

Olga Cruz-Lopez

3

1 reference

5 August 2017

Ernest Hamel

10

1 reference

5 August 2017

language of work or name

English

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publication date

21 November 2010

1 reference

Bioorganic & Medicinal Chemistry Letters

5 August 2017

published in

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5 August 2017

volume

21

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5 August 2017

issue

9

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5 August 2017

page(s)

2746-2751

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Tubulin-interactive natural products as anticancer agents

5 August 2017

cites work

1 reference

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Synthesis and biological evaluation of 1-methyl-2-(3',4',5'-trimethoxybenzoyl)-3-aminoindoles as a new class of antimitotic agents and tubulin inhibitors

8 July 2018

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8 July 2018

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8 July 2018

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Synthesis and biological evaluation of 2-amino-3-(3',4',5'-trimethoxybenzoyl)-5-aryl thiophenes as a new class of potent antitubulin agents

8 July 2018

1 reference

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Medicinal chemistry of combretastatin A4: present and future directions.

8 July 2018

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8 July 2018

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8 July 2018

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Review: tubulin function, action of antitubulin drugs, and new drug development

8 July 2018

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8 July 2018

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Structural requirements for the interaction of combretastatins with tubulin: how important is the trimethoxy unit?

8 July 2018

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Combretastatin A-4 analogues as antimitotic antitumor agents

8 July 2018

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Evaluation of antimitotic agents by quantitative comparisons of their effects on the polymerization of purified tubulin

8 July 2018

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Microtubule dynamics and tubulin interacting proteins

8 July 2018

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Antineoplastic agents. 379. Synthesis of phenstatin phosphate

8 July 2018

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Isolation and structure of the strong cell growth and tubulin inhibitor combretastatin A-4.

8 July 2018

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Human chronic myelogenous leukemia cell-line with positive Philadelphia chromosome

8 July 2018

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Microtubule structure and its stabilisation

8 July 2018

1 reference

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Synthesis and structure-activity relationship of 2-aminobenzophenone derivatives as antimitotic agents.

26 October 2018

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Structure-activity analysis of the interaction of curacin A, the potent colchicine site antimitotic agent, with tubulin and effects of analogs on the growth of MCF-7 breast cancer cells.

26 October 2018

1 reference

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Synthesis and evaluation of analogs of (Z)-1-(4-methoxyphenyl)-2-(3,4,5-trimethoxyphenyl)ethene as potential cytotoxic and antimitotic agents

26 October 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/21146985

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Antimitotic natural products combretastatin A-4 and combretastatin A-2: studies on the mechanism of their inhibition of the binding of colchicine to tubulin

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/21146985

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1016/J.BMCL.2010.11.083

1 reference

5 August 2017

1 reference

5 August 2017

1 reference