Identification of the hydrophobic ligand binding pocket of the S1P1 receptor (Q33264060)

24 July 2017

title

Identification of the hydrophobic ligand binding pocket of the S1P1 receptor (English)

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24 July 2017

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Karoly Liliom

6

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author name string

Yuko Fujiwara

1

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24 July 2017

Daniel A Osborne

2

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24 July 2017

Michelle D Walker

3

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24 July 2017

De-an Wang

4

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24 July 2017

Debra A Bautista

5

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24 July 2017

James R Van Brocklyn

7

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24 July 2017

Abby L Parrill

8

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24 July 2017

Gabor Tigyi

9

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24 July 2017

language of work or name

English

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publication date

18 November 2006

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Journal of Biological Chemistry

24 July 2017

published in

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24 July 2017

volume

282

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24 July 2017

issue

4

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24 July 2017

page(s)

2374-2385

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S1P1-selective in vivo-active agonists from high-throughput screening: off-the-shelf chemical probes of receptor interactions, signaling, and fate

24 July 2017

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21 June 2018

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21 June 2018

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21 June 2018

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Alteration of lymphocyte trafficking by sphingosine-1-phosphate receptor agonists

21 June 2018

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Identification by site-directed mutagenesis of residues involved in ligand recognition and activation of the human A3 adenosine receptor

21 June 2018

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A single amino acid determines lysophospholipid specificity of the S1P1 (EDG1) and LPA1 (EDG2) phospholipid growth factor receptors

21 June 2018

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21 June 2018

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21 June 2018

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Edg-1, the G protein-coupled receptor for sphingosine-1-phosphate, is essential for vascular maturation

21 June 2018

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Identification of Edg1 receptor residues that recognize sphingosine 1-phosphate.

21 June 2018

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A sphingosine-1-phosphate receptor regulates cell migration during vertebrate heart development

21 June 2018

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21 June 2018

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Sphingosine 1-phosphate regulates melanoma cell motility through a receptor-coupled extracellular action and in a pertussis toxin-insensitive manner

21 June 2018

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21 June 2018

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21 June 2018

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21 June 2018

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21 January 2018

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21 January 2018

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21 January 2018

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Protein kinase C epsilon dependence of the recovery from down-regulation of S1P1 G protein-coupled receptors of T lymphocytes

21 January 2018

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21 January 2018

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Site-directed mutagenesis at the human B2 receptor and molecular modelling to define the pharmacophore of non-peptide bradykinin receptor antagonists

21 January 2018

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The biologically crucial C terminus of cholecystokinin and the non-peptide agonist SR-146,131 share a common binding site in the human CCK1 receptor. Evidence for a crucial role of Met-121 in the activation process

21 January 2018

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Role of charged amino acids conserved in the vasoactive intestinal polypeptide/secretin family of receptors on the secretin receptor functionality

21 January 2018

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PubMed

https://pubmed.ncbi.nlm.nih.gov/17114791

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

CCK-B/Gastrin receptor transmembrane domain mutations selectively alter synthetic agonist efficacy without affecting the activity of endogenous peptides

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/17114791

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1074/JBC.M609648200

1 reference

24 July 2017

1 reference

24 July 2017

1 reference