Benzodiazepines and benzotriazepines as protein interaction inhibitors targeting bromodomains of the BET family (Q27675927)

2

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Panagis Filippakopoulos

1

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Oleg Fedorov

Oleg Fedorov

3

0 references

Stefan Knapp

Stefan Knapp

8

0 references

Olaf Morgenstern

6

Olaf Morgenstern

0 references

Franz Bracher

7

Franz Bracher

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author name string

Marco Keller

4

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Matthias Wrobel

Bioorganic & Medicinal Chemistry

5

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language of work or name

English

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publication date

15 March 2012

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published in

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volume

20

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issue

6

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page(s)

1878-86

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cites work

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Expression of BRD7-interacting proteins,BRD2 and BRD3, in nasopharyngeal carcinoma tissues

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BRD4-NUT fusion oncogene: a novel mechanism in aggressive carcinoma

20 March 2017

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RNAi screen identifies Brd4 as a therapeutic target in acute myeloid leukaemia

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Flavopiridol induces BCL-2 expression and represses oncogenic transcription factors in leukemic blasts from adults with refractory acute myeloid leukemia

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29 September 2017

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29 September 2017

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29 September 2017

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29 September 2017

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The separation of 3H-Benzodiazepine binding sites in brain and of benzodiazepine pharmacological properties

29 September 2017

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6-Phenyl-4H-s-triazolo[4,3-a][1,4]benzodiazepines which have central nervous system depressant activity

29 September 2017

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29 September 2017

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2 June 2018

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A novel indazolo-triazolo-benzotriazepine exerts anti-inflammatory effects by inhibition of cyclooxygenase-2 activity and nitric oxide synthase-2 expression.

2 June 2018

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10.1016/J.BMC.2011.10.080

27 November 2018

Identifiers

DOI

1 reference

1 reference

1 reference

PubMed publication ID

22137933

1 reference