(Q39648105)

13 September 2017

Impact of linker length on the activity of PROTACs (English)

1 reference

13 September 2017

Kedra Cyrus

1

1 reference

13 September 2017

Marie Wehenkel

2

1 reference

13 September 2017

Eun-Young Choi

3

1 reference

13 September 2017

Hyeong-Jun Han

4

1 reference

13 September 2017

Hyosung Lee

5

1 reference

13 September 2017

Hollie Swanson

6

1 reference

13 September 2017

Kyung-Bo Kim

7

1 reference

13 September 2017

4 October 2010

1 reference

13 September 2017

1 reference

13 September 2017

7

1 reference

13 September 2017

2

1 reference

13 September 2017

359-364

1 reference

Protein knockdown using methyl bestatin-ligand hybrid molecules: design and synthesis of inducers of ubiquitination-mediated degradation of cellular retinoic acid-binding proteins.

13 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3835402

Chemical inducers of targeted protein degradation

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3835402

Design and Applications of Bifunctional Small Molecules: Why Two Heads Are Better Than One.

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3835402

Discovery and development of heat shock protein 90 inhibitors

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3835402

The ubiquitin system, disease, and drug discovery

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3835402

To ubiquitinate or to deubiquitinate: it all depends on the partners

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3835402

Targeted intracellular protein degradation induced by a small molecule: En route to chemical proteomics

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3835402

From Knowing to Controlling: A Path from Genomics to Drugs Using Small Molecule Probes

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3835402

Protacs: chimeric molecules that target proteins to the Skp1-Cullin-F box complex for ubiquitination and degradation

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3835402

SCF and Cullin/Ring H2-based ubiquitin ligases

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3835402

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3835402

Targeting steroid hormone receptors for ubiquitination and degradation in breast and prostate cancer

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3835402

Chimeric molecules to target proteins for ubiquitination and degradation

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3835402

Chemical genetic control of protein levels: selective in vivo targeted degradation

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3835402

Deciphering isozyme function: exploring cell biology with chemistry in the post-genomic era.

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3835402

Targeted Degradation of Proteins by PROTACs.

25 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3835402

Development of an aryl hydrocarbon receptor antagonist using the proteolysis-targeting chimeric molecules approach: a potential tool for chemoprevention

21 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3835402

Synthesis of chimeric 7alpha-substituted estradiol derivatives linked to cholesterol and cholesterylamine.

21 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3835402

Synthesis and evaluation of hexahydrochrysene and tetrahydrobenzofluorene ligands for the estrogen receptor

21 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3835402

The estrogen receptor: a structure-based approach to the design of new specific hormone-receptor combinations.

21 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3835402

Synthesis and evaluation of geldanamycin-estradiol hybrids

21 August 2018

1 reference

https://pubmed.ncbi.nlm.nih.gov/20922213

12 December 2020

Identification of a geldanamycin dimer that induces the selective degradation of HER-family tyrosine kinases

1 reference

https://pubmed.ncbi.nlm.nih.gov/20922213

12 December 2020

Degradation of target protein in living cells by small-molecule proteolysis inducer

1 reference

https://pubmed.ncbi.nlm.nih.gov/20922213

12 December 2020

Targeted degradation of the aryl hydrocarbon receptor by the PROTAC approach: a useful chemical genetic tool

1 reference

https://pubmed.ncbi.nlm.nih.gov/20922213

12 December 2020

Synthesis and evaluation of geldanamycin-testosterone hybrids

1 reference

https://pubmed.ncbi.nlm.nih.gov/20922213

12 December 2020

Identifiers

DOI

10.1039/C0MB00074D

1 reference

13 September 2017

1 reference

13 September 2017

PubMed publication ID

20922213

1 reference