Selleck Screening Libraries offer easy,

ready-to-use alternatives for the analysis

of biochemical pathways and pharmaceutical-
related applications. Our library contains a
unique and diverse collection of over 700
bioactive compounds suitable for high-
throughput screening (HTS), cell based
high-content screening (HCS), chemical and
biological applications.
Library Advantages
Selleck Screening Libraries
Structurally diverse, medicinally active and cell permeable
Rich documentation with structure, IC50 and customer reviews
NMR and HPLC to ensure the high purity
The collection of unique small molecules is focused
on over 200 targets in more than 20 signaling
pathways, such as PI3K / mTOR / Akt, MAPK
and apoptosis. We provide compound position
information, physical information, biological activity
and chemical properties for each plate.
www.selleckchem.com/screening/screening-library.html
Chemical Library Total
A collection of 712 bioactive compounds.
Inhibitor Library
A collection of 335 inhibitors.
Kinase Inhibitor Library
A collection of 150 kinase inhibitors.
FDA Approved Drug Library
A collection of 381 FDA approved drugs.
Natural Product Library
A collection of 130 natural products.
Chemotherapeutic Agent Library
A collection of 40 chemotherapeutic agents.
Tyrosine Kinase Inhibitor Library
A unique collection of 86 tyrosine kinase inhibitors.
Chemical Library Total (96-well)
Chemical Library Total
l
Toll Free:(877)796-6397 www.selleckchem.com [email protected]
Phone:+1-832-582-8158
---USA and Canada only---
A unique collection of 712 bioactive compounds for high throughput screening (HTS)
and high content screening (HCS)
Bioactivity and safety confirmed by preclinical research and clinical trials
Some compounds have been approved by FDA
Includes most Selleck inhibitors, APIs, natural products and chemotherapeutic agents
Structurally diverse, medicinally active and cell permeable
Rich documentation with structure, IC50 and customer reviews
NMR and HPLC to ensure the high purity
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Chemical Library Total
Product
712
Compounds
L1700
Catalog No.
Powder Pre-dissolved in DMSO
Size
You can select compounds, quantities, formatGU\VROLGRU'062plate map and concentration
to meet your specific requirement.
Customize Your Library
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100
200
400
300
Inhibitors Kinase Inhibitors FDA Approved Drugs Natural Products Chemotherapeutic Agents
335
150
381
130
40
Tyrosine Kinase Inhibitors
86
Download the Library Total
SDF
Download the Library Total
XLSX
ww.selleckchem.com
Download
SDF
SDF
Download comprehensive documentation on this library:
Inhibitor Library
Terrific Quality, Validation, Customer Review & Tech Support
2
Inhibitor Library (96-well)
A unique collection of 335 inhibitors for high throughput screening (HTS) and high content
screening (HCS)
Bioactivity and safety confirmed by preclinical research and clinical trials
Some inhibitors have been approved by FDA
Structurally diverse, medicinally active and cell permeable
Rich documentation with structure, IC50 and customer reviews
NMR and HPLC to ensure the high purity
Targets PI3K, VEGFR and RTK pathway, HDAC, Aurora Kinase, CDK and Cell Cycle regulators,
Integrase/Proteasome etc
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to meet your specific requirement.
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Inhibitor Library 335 L1100
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Powder Pre-dissolved in DMSO
Size
18
11
3 3
1
1 1 1 1 1 1 1 1 1 1 1 1 1 1
1
2
2 2 2 2 2 2 2 2
27
16 16
15
14 14
11
7 7
1
8 8
4
4 4 4
2 2
12 12
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3
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7 7
4 4
2 2
11
5
5 5
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6 6 6
6 6 6
31
9 9 9
10
0
2
4
6
8
10
12
14
16
18
20
22
24
26
28
30
32
0
2
4
6
8
10
PI3K
mTOR
AKT
GSK-3
DNA-PK
$70
S6 kinase
VEGFR
EGFR
PDGFR
c-Kit
F0HW
Bcr-Abl
SRC
IGF-1R
HER2
ALK
Syk
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FGFR
HIF
VDA
Bcl-2
TNF-alpha
p53
Survivin
JAK
STAT
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Kinesin Spindle Protein
Aurora Kinase
HDAC HSP
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Sirtuin
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PARP
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Dihydrofolate Reductas
5-HT receptor
COX
Histamine
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Gamma-secretase
mAChRs
GABA
receptor
Dopamine Receptor
Hedgehog
Wnt
Adrenergic
Receptors
ETA-receptor
5-alpha-reductase
Estrogen Receptor
Androgen
Receptor
RAAS
Aromatase
Calcium
Channel
Sodium Channel
Potassium
Channel
P450
Factor Xa
PDE
Aminopeptidase
Dehydrogenase
Proteasome
HCV
Protease
DPP-4
HIV Protease
CCR5
Reverse
Transcriptase
CFTR
Integrase
Others
Download the Inhibitor Library
SDF
Download the Inhibitor Library
XLSX
Terr
2
Download
SDF
SDF
Download comprehensive documentation on this library:
Kinase Inhibitor Library (96-well)
Kinase Inhibitor Library
3
Toll Free:(877)796-6397 www.selleckchem.com [email protected]
Phone:+1-832-582-8158
---USA and Canada only---
A unique collection of 150 kinase inhibitors for high throughput screening (HTS) and
high content screening (HCS)
Bioactivity and safety confirmed by preclinical research and clinical trials
Some kinase inhibitors have been approved by FDA
Targets kinases such as RTKs, PI3K, Aurora Kinase, CDK and MEK
Most are ATP competitive
Structurally diverse, medicinally active and cell permeable
Rich documentation with structure, IC50 and customer reviews
NMR and HPLC to ensure the high purity
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to meet your specific requirement.
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Powder Pre-dissolved in DMSO
Size
18
28
11
3 3
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15
14
4
11 11
7 7
10 10
8
2 2
12
15
6 6 6
8
2
44
2 2
1 1 1 1
0
2
4
6
8
10
12
14
16
18
20
22
24
26
28
PI3K
mTOR
AKT
GSK-3
$70
VEGFR
EGFR
PDGFR
JAK
0(.
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c-Kit
F0HW
Bcr-Abl
SRC
IGF-1R
HER2
ALK
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FGFR
Aurora
CDK
PLK
PKC
S6 Kinase
TGF-beta
CHK
JNK
Others
Download the Kinase Inhibitor
Library SDF
Download the Kinase Inhibitor
Library XLSX
www.selleckchem.co
Download
Library SD
SDF
Download comprehensive documentation on this library:
Tyrosine Kinase Inhibitor Library (96-well)
A unique collection of 86 tyrosine kinase inhibitors for high throughput screening (HTS)
and high content screening (HCS)
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Tyrosine Kinase
Inhibitor Library
86 L1800
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Powder Pre-dissolved in DMSO
Size
Terrific Quality, Validation, Customer Review & Tech Support
4
Bioactivity and safety confirmed by preclinical research and clinical trials
Some tyrosine kinase inhibitors have been approved by FDA
Targets tyrosine kinases such as EGFR, VEGFR, SRC, c-Met and JAK
Structurally diverse, medicinally active and cell permeable
Rich documentation with structure, IC50 and customer reviews
NMR and HPLC to ensure the high purity
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VEGFR EGFR PDGFR JAK Raf c-Kit F0HW Bcr-Abl IGF-1R HER2 ALK Syk SRC Tie2 )OW)/. FGFR Wee1
Download the Tyrosine Kinase
Inhibitor Library SDF
Download the Tyrosine Kinase
Inhibitor Library XLSX
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Download
Inhibitor Li
SDF
Download comprehensive documentation on this library:
FDA Approved Drug Library
FDA Approved Drug Library (96-well)
A unique collection of 381 FDA approved drugs for high throughput screening (HTS) and
high content screening (HCS)
Helps to locate new targets for old drugs
Bioactivity and safety confirmed by clinical trials
All compounds have been approved by FDA
Structurally diverse, medicinally active and cell permeable
Rich documentation with structure, IC50 and customer reviews
NMR and HPLC to ensure the high purity
Related to oncology, cardiology, anti-inflammatory, immunology, neuropsychiatry,
analgesia etc
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to meet your specific requirement.
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FDA Approved
Drug Library
381 L1300
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0
10
20
30
40
50
60
70
80
65
77
40
25
31
20
69
59
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Cancer
Infection
Endocrinology
0HWDEROLF
Disease
Inflammation
Immunology
Neurological
Disease
Cardiovascular
Disease
Respiratory
Diseases
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Toll Free:(877)796-6397 www.selleckchem.com [email protected]
Phone:+1-832-582-8158
---USA and Canada only---
Download the FDA Approved
Drug Library SDF
Download the FDA Approved
Drug Library XLSX
www.selleckchem.co
Download
Drug Libra
SDF
Download comprehensive documentation on this library:
Natural Product Library (96-well)
Natural Product Library
A unique collection of 130 natural products for high throughput screening (HTS) and
high content screening (HCS)
Structurally diverse, bioactive and cell permeable
Rich documentation with structure and IC50
NMR and HPLC to ensure the high purity
Library includes:
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to meet your specific requirement.
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Natural Product Library 130 L1400
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Product Compounds Catalog No.
Powder Pre-dissolved in DMSO
Size
Steroid saponins
Benzoquinones
Tannins
Alkaloids
PPGs
Penzaldehydes
Saccharides
Anthraquinones
Phenanthraquinones
Phenylcarbinols
Pyrimidines
Flavones
Synthetic derivatives
Phenethylamines
Acid amides
Steroids
Peptides
Terrific Quality, Validation, Customer Review & Tech Support
6
Download the Natural Product
Library XLSX
Download the Natural Product
Library SDF
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Download
Library SD
SDF
Download comprehensive documentation on this library:
Chemotherapeutic Agent Library
Chemotherapeutic Agent Library (96-well)
A unique collection of 40 chemotherapeutic agents for high throughput screening (HTS)
and high content screening (HCS)
Structurally diverse, medicinally active and cell permeable
Rich documentation with structure, IC50 and customer reviews
NMR and HPLC to ensure the high purity
Bioactivity and safety confirmed by clinical trials
Some agents have been approved by FDA for both oncological and non-oncological purposes
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Chemotherapeutic
Agent Library
40 L1500
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Powder Pre-dissolved in DMSO
Size
0
2
4
6
8
10
12
14
6
13
3
4 4
10
Alkylating
agents
Anti-metabolites
Plant alkaloids
and terpenoids
Topoisomerase
inhibitors
Cytotoxic
antibiotics
Other antitumour
agents
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Toll Free:(877)796-6397 www.selleckchem.com [email protected]
Phone:+1-832-582-8158
---USA and Canada only---
Download the Chemotherapeutic
Agent Library XLSX
Download the Chemotherapeutic
Agent Library SDF
www.selleckchem.co
Download th
Agent Librar
SDF
Download comprehensive documentation on this library:
Guaranteed Quality and Support
Guaranteed Quality and Support
The purity of each reagent in Selleck screening libraries is confirmed by HPLC
and H-NMR.
In addition, all libraries are supplied with a detailed documentation set including
compound position information, physical information, biological activity and
chemical properties in SDF and Excel files.
Certificate of Analysis
Molecular Formula: C
17
H
15
BrClFN
4
O
3
Molecular Weight: 457.68
CAS No.: 606143-52-6
Storage: at -20 2 years
Molecular Structure:
AU
0.00
0.50
1.00
1.50
2.00
2.50
3.00
0inutes
2.00 4.00 6.00 8.00 10.00 12.00 14.00 16.00 18.00 20.00 22.00 24.00 26.00 28.00 30.00
1
5
.6
7
6
1
6
.1
5
2
1
7
.8
7
5
11.693
8.379
7.892
7.722
7.589
7.587
7.584
7.581
7.252
7.251
7.247
7.230
7.228
7.225
6.353
6.343
6.331
6.321
4.694
4.691
3.882
3.839
3.533
3.311
3.309
2.483
2.479
2.476
2.475
2.063
2.059
-0.025
-0.028
1.00
0.96
1.00 0.94 1.00 3.01
2.00
2.00 1.00 1.00
0.91
12 10 8 6 4 2 0 330
6'062G
HN
Cl
Br F N
N
HN O O HO
USER: -- DATE: Apr 2 2011
Nuts - $S100810 AZD6244
Std proton;blank line
8 6 7 2 3 , 1 2 5 6 1 : d 1 S T P 4 . 4 1 2 3 : 1 F O 5 6 0 8 : 1 W S 7 9 4 . 0 0 1 : 2 F 5 3 6 . 9 9 3 : 1 F
0 . 0 : B L 8 : A N c e s 0 . 2 : D P s u 2 . 7 : W P l u p 2 s : X E
Physical and chemical properties
S1008 AZD6244 (Selumetinib)
SD File
XLSX File
Having doubts on Sellecks products?
Following data from our customers is to assure you the high quality of Selleck Screening Libraries.
Data from [ Nature Biotechnology0DUFK@
Vorinostat (SAHA) purchased from Selleck
Data from [ Cancer Cell-XQH@
Rapamycin (Sirolimus) purchased from Selleck
Data from [ Nature1RYHPEHU@
AZD6244 (Selumetinib) purchased from Selleck
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Customize Your Library
Customize Your Library
A cherry pick service is available to let you customize your own libraries.
Please contact us at [email protected] to check the details of your library.
You could select
Specific Compounds
Quantities
Format GU\VROLGRU'062VROXWLRQ
Plate map
Concentration
9
Toll Free:(877)796-6397 www.selleckchem.com [email protected]
Phone:+1-832-582-8158
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Tel:
Web:
Russia
COPRAS
Email:
+74 953331163
www.copras.ch
[email protected]
Australia
Life Research Pty Ltd
Tel:
Email:
Web:
+61 398030045
[email protected]
www.liferesearch.com
Austria
eubio
Tel:
Email:
Web:
+43 18950145
[email protected]
www.eubio.at
Canada
Cedarlane
Tel:
Email:
Web:
+1 289 288 0001
[email protected]
www.cedarlanelabs.com
China
BinXin Bio, Co Ltd
Tel:
Email:
Web:
+86 22 23915166
[email protected]
[email protected]
China
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Divbio Science
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Absource Diagnostics GmbH
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Germany
ICS International Clinical Service GmbH
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Japan
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Aurogene
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COSMO BIO CO., LTD
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Wako Pure Chemical Industries, Ltd.
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RUSCHEMBIO
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VWR International LLC
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UK
Stratech Scientific Ltd.
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Lumtec
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