Molecular imaging of lymphoid organs and immune activation by positron emission tomography with a new [18F]-labeled 2'-deoxycytidine analog

Nat Med. 2008 Jul;14(7):783-8. doi: 10.1038/nm1724. Epub 2008 Jun 8.

Abstract

Monitoring immune function with molecular imaging could have a considerable impact on the diagnosis and treatment evaluation of immunological disorders and therapeutic immune responses. Positron emission tomography (PET) is a molecular imaging modality with applications in cancer and other diseases. PET studies of immune function have been limited by a lack of specialized probes. We identified [(18)F]FAC (1-(2'-deoxy-2'-[(18)F]fluoroarabinofuranosyl) cytosine) by differential screening as a new PET probe for the deoxyribonucleotide salvage pathway. [(18)F]FAC enabled visualization of lymphoid organs and was sensitive to localized immune activation in a mouse model of antitumor immunity. [(18)F]FAC microPET also detected early changes in lymphoid mass in systemic autoimmunity and allowed evaluation of immunosuppressive therapy. These data support the use of [(18)F]FAC PET for immune monitoring and suggest a wide range of clinical applications in immune disorders and in certain types of cancer.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Animals
  • Deoxycytidine / analogs & derivatives*
  • Deoxycytidine / chemistry
  • Fluorine Radioisotopes*
  • Fluorodeoxyglucose F18
  • Lymphoscintigraphy*
  • Mice
  • Mice, Inbred C57BL
  • Mice, Inbred MRL lpr
  • Positron-Emission Tomography / methods*
  • Radionuclide Imaging / methods*
  • Radiopharmaceuticals
  • Sensitivity and Specificity
  • Tissue Distribution

Substances

  • Fluorine Radioisotopes
  • Radiopharmaceuticals
  • Deoxycytidine
  • Fluorodeoxyglucose F18