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|---|---|
| Systematic (IUPAC) name | |
| 1-(4-fluorophenyl)-4-(4-pyridin-2-ylpiperazin-1-yl)butan-1-one | |
| Clinical data | |
| AHFS/Drugs.com | International Drug Names |
| Pregnancy cat. | ? |
| Legal status | ? |
| Routes | intramuscular injection |
| Pharmacokinetic data | |
| Metabolism | hepatic |
| Half-life | 4 hours |
| Identifiers | |
| CAS number | 1649-18-9  |
| ATCvet code | QN01AX91 QN05AD90 |
| PubChem | CID 15443 |
| ChemSpider | 14695  |
| UNII | 19BV78AK7W |
| KEGG | D02620 |
| ChEMBL | CHEMBL340211 |
| Chemical data | |
| Formula | C19H22FN3O |
| Mol. mass | 327.396 g/mol |
| SMILES | eMolecules & PubChem |
|
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| Physical data | |
| Melt. point | 90–95 °C (194–203 °F) |
 (what is this?) (verify) |
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Azaperone (Stresnil, Fluoperidol) is a pyridinylpiperazine and butyrophenone neuroleptic drug with sedative and antiemetic effects, which is used mainly as a tranquilizer in veterinary medicine. It is used mainly in pigs and elephants. [1] More rarely it may be used in humans as an antipsychotic drug, but this is uncommon. Use in horses is avoided as adverse reactions may occur.
Azaperone acts primarily as a dopamine antagonist but also has some antihistaminic and anticholinergic properties as seen with similar drugs such as haloperidol. Azaperone may cause hypotension and while it has minimal effects on respiration in pigs, high doses in humans can cause respiratory depression which may be why it is rarely used in humans.
The most common use for azaperone is in relatively small doses to reduce aggression in farmed pigs, either to stop them fighting or to encourage sows to accept piglets. Higher doses are used for anesthesia in combination with other drugs such as xylazine, tiletamine and zolazepam. Azaperone is also used in combination with strong narcotics such as etorphine or carfentanil for tranquilizing large animals such as elephants.
References [link]
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https://wn.com/Azaperone
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Eyesburn
by: EyesburnSo much trouble in the world
So much trouble in the world
Bless my eyes this morning
Jah sun is on the rise once again
The way earthly thin's are goin'
Anything can happen.
You see men sailing on their ego trips,
Blast off on their space ships,
Million miles from reality:
No care for you, no care for me.
So much trouble in the world;
So much trouble in the world.
All you gotta do: Give a little (give a little),
take a little (take a little), give a little (give a little)!
One more time, ye-ah! (give a little) Ye-ah! (take a little)
Ye-ah! (give a little) Yeah!
So you think you've found the solution,
But it's just another illusion!
(So before you check out this tide),
Don't leave another cornerstone
Standing there behind, eh-eh-eh-eh!
We've got to face the day;
(Ooh) Ooh-wee, come what may:
We the street people talkin',
Yeah, we the people strugglin'.
Now they sitting on a time bomb; (Bomb-bomb-bomb! Bomb-bomb-bomb!)
Now I know the time has come: (Bomb-bomb-bomb! Bomb-bomb-bomb!)
What goes on up is coming on down, (Bomb-bomb-bomb! Bomb-bomb-bomb!)
Goes around and comes around. (Bomb-bomb-bomb! Bomb-bomb-bomb!)
So much trouble in the world;
So much trouble in the world;
So much trouble in the world.
There is so much trouble (so much trouble in the world);
There is so much trouble;
There is so much trouble (so much in the world);
There is so much trouble;
There is so much trouble in the world (so much trouble in the world);
There is (so much in the world);