LRRK2 Regulates CPT1A to Promote β-Oxidation in HepG2 Cells

Molecules. 2020 Sep 9;25(18):4122. doi: 10.3390/molecules25184122.

Abstract

Leucine-rich repeat kinase 2 (LRRK2) is involved in lipid metabolism; however, the role of LRRK2 in lipid metabolism to affect non-alcoholic fatty liver disease (NAFLD) is still unclear. In the mouse model of NAFLD induced by a high-fat diet, we observed that LRRK2 was decreased in livers. In HepG2 cells, exposure to palmitic acid (PA) down-regulated LRRK2. Overexpression and knockdown of LRRK2 in HepG2 cells were performed to further investigate the roles of LRRK2 in lipid metabolism. Our results showed that β-oxidation in HepG2 cells was promoted by LRRK2 overexpression, whereas LRRK2 knockdown inhibited β-oxidation. The critical enzyme of β-oxidation, carnitine palmitoyltransferase 1A (CPT1A), was positively regulated by LRRK2. Our data suggested that the regulation of CPT1A by LRRK2 may be via the activation of AMP-activated protein kinase (AMPK) and peroxisome proliferator-activated receptor α (PPARα). The overexpression of LRRK2 reduced the concentration of a pro-inflammatory cytokine, tumor necrosis factor α (TNFα), induced by PA. The increase in β-oxidation may promote lipid catabolism to suppress inflammation induced by PA. These results indicated that LRRK2 participated in the regulation of β-oxidation and suggested that the decreased LRRK2 may promote inflammation by suppressing β-oxidation in the liver.

Keywords: CPT1A; LRRK2; NAFLD; β-oxidation.

MeSH terms

  • Animals
  • Carnitine O-Palmitoyltransferase / physiology*
  • Cell Nucleus / metabolism
  • Cytokines / metabolism
  • Diet, High-Fat
  • Hep G2 Cells
  • Humans
  • Inflammation
  • Leucine-Rich Repeat Serine-Threonine Protein Kinase-2 / physiology*
  • Lipid Metabolism
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Non-alcoholic Fatty Liver Disease / metabolism
  • Oxidation-Reduction
  • Oxygen / metabolism*
  • PPAR alpha / metabolism
  • Palmitic Acid / pharmacology
  • Tumor Necrosis Factor-alpha / metabolism

Substances

  • Cytokines
  • PPAR alpha
  • Tumor Necrosis Factor-alpha
  • Palmitic Acid
  • CPT1A protein, human
  • CPT1B protein, mouse
  • Carnitine O-Palmitoyltransferase
  • LRRK2 protein, human
  • Leucine-Rich Repeat Serine-Threonine Protein Kinase-2
  • Lrrk2 protein, mouse
  • Oxygen