N-acetyl cysteine mediates protection from 2-hydroxyethyl methacrylate induced apoptosis via nuclear factor kappa B-dependent and independent pathways: potential involvement of JNK

Toxicol Sci. 2009 Apr;108(2):356-66. doi: 10.1093/toxsci/kfp010. Epub 2009 Jan 28.

Abstract

The mechanisms by which resin based materials induce adverse effects in patients have not been completely elucidated. Here we show that 2-hydroxyethyl methacrylate (HEMA) induces apoptotic cell death in oral keratinocytes. Functional loss and cell death induced by HEMA was significantly inhibited in the presence of N-acetyl cysteine (NAC) treatment. NAC also prevented HEMA mediated decrease in vascular endothelial growth factor secretion. The protective effect of NAC was partly related to its ability to induce NF-kappaB in the cells, since HEMA mediated inhibition of nuclear NF-kappaB expression and function was significantly blocked in the presence of NAC treatment. Moreover, blocking of nuclear translocation of NF-kappaB in oral keratinocytes sensitized these cells to HEMA mediated apoptosis. In addition, since NAC was capable of rescuing close to 50% of NF-kappaB knockdown cells from HEMA mediated cell death, there is, therefore, an NF-kappaB independent pathway of protection from HEMA mediated cell death by NAC. NAC mediated prevention of HEMA induced cell death in NF-kappaB knockdown cells was correlated with a decreased induction of c-Jun N-terminal kinase (JNK) activity since NAC inhibited HEMA mediated increase in JNK levels. Furthermore, the addition of a pharmacologic JNK inhibitor to HEMA treated cells prevented cell death and restored NF-kappaB knockdown cell function significantly. Therefore, NAC protects oral keratinocytes from the toxic effects of HEMA through NF-kappaB dependent and independent pathways. Moreover, our data suggest the potential involvement of JNK pathway in NAC mediated protection.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Acetylcysteine / pharmacology*
  • Apoptosis / drug effects*
  • Blotting, Western
  • Cell Line
  • Cell Nucleus / drug effects
  • Cytokines / biosynthesis
  • Cytoplasm / drug effects
  • Cytoplasm / metabolism
  • DNA / biosynthesis
  • DNA / genetics
  • Dental Materials / toxicity*
  • Enzyme Activation / drug effects
  • Enzyme-Linked Immunosorbent Assay
  • Free Radical Scavengers / pharmacology*
  • Gene Transfer Techniques
  • Humans
  • JNK Mitogen-Activated Protein Kinases / physiology*
  • Keratinocytes / drug effects
  • Luciferases / metabolism
  • Methacrylates / toxicity*
  • NF-kappa B / antagonists & inhibitors*
  • NF-kappa B / physiology*
  • Retroviridae / genetics
  • Signal Transduction / drug effects

Substances

  • Cytokines
  • Dental Materials
  • Free Radical Scavengers
  • Methacrylates
  • NF-kappa B
  • hydroxyethyl methacrylate
  • DNA
  • Luciferases
  • JNK Mitogen-Activated Protein Kinases
  • Acetylcysteine