(Q56028298)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:33398642%20AND%20SRC:MED&resulttype=core&format=json

9 January 2021

author name string

Aliya Ibrar

series ordinal

2

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:33398642%20AND%20SRC:MED&resulttype=core&format=json

9 January 2021

Sumera Zaib

series ordinal

3

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:33398642%20AND%20SRC:MED&resulttype=core&format=json

Topics in Current Chemistry

9 January 2021

publication date

January 1975

0 references

published in

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:33398642%20AND%20SRC:MED&resulttype=core&format=json

9 January 2021

volume

379

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:33398642%20AND%20SRC:MED&resulttype=core&format=json

9 January 2021

issue

1

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:33398642%20AND%20SRC:MED&resulttype=core&format=json

9 January 2021

page(s)

3

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:33398642%20AND%20SRC:MED&resulttype=core&format=json

The Substitution of Aryl Iodides with Cuprous Acetylides. A Synthesis of Tolanes and Heterocyclics1

9 January 2021

cites work

1 reference

Crossref

https://api.crossref.org/works/10.1016%2FS0040-4039%2800%2991094-3

7 January 2021

inferred from DOI database lookup

Synthesis of aryl- and vinyl-substituted acetylene derivatives by the use of nickel and palladium complexes

1 reference

Crossref

https://api.crossref.org/works/10.1016%2FS0040-4039%2800%2991094-3

7 January 2021

inferred from DOI database lookup

Palladium catalyzed synthesis of aryl, heterocyclic and vinylic acetylene derivatives

1 reference

Crossref

https://api.crossref.org/works/10.1016%2FS0040-4039%2800%2991094-3

7 January 2021

inferred from DOI database lookup

Correlation of biological activity and high-pressure liquid chromatographic retention index for a series of propranolol, barbiturate, and anthranilic acid analogs

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Benzodiazepine receptor binding of nonbenzodiazepines in vivo: alpidem, zolpidem and zopiclone

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

New 5H-pyridazino[4,5-b]indole derivatives. Synthesis and studies as inhibitors of blood platelet aggregation and inotropics.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Design of enzyme inhibitors using iterative protein crystallographic analysis

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis of 11-phenyl-2,3,4,5-tetrahydro-1H-(1,4)diazepino(1,2-a)indoles and 1-(3-aminopropyl)-2-hydroxymethyl-3-phenylindoles as 5-hydroxytryptamine antagonists

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Immunopharmacological studies on TBX, a new antiallergic drug (1). Inhibitory effects on passive cutaneous anaphylaxis in rats and guinea pigs

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Microsomal metabolism of pyrrolizidine alkaloids from Senecio jacobaea. Isolation and quantification of 6,7-dihydro-7-hydroxy-1-hydroxymethyl-5H-pyrrolizine and N-oxides by high performance liquid chromatography

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Cytotoxicity of sesquiterpene lactones.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Two dihydropyrrolizine alkaloid metabolites isolated from mouse hepatic microsomes in vitro

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Debrisoquine-type polymorphism of drug oxidation: purification from human liver of a cytochrome P450 isozyme with high activity for bufuralol hydroxylation

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis and assembly of membrane glycoproteins. Membrane anchoring COOH-terminal domain of vesicular stomatitis virus envelope glycoprotein G contains fatty acids

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

The type I insulin-like growth factor receptor mediates the rapid effects of multiplication-stimulating activity on membrane transport systems in rat soleus muscle

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Neurochemical and behavioral evidence that quipazine-ketanserin discrimination is mediated by serotonin2A receptor.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

[[[(Thienylcarbonyl)alkyl]oxy]phenyl]- and [[[(pyrrylcarbonyl)alkyl]oxy]phenyl]oxazoline derivatives with potent and selective antihuman rhinovirus activity.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

A new series of PDGF receptor tyrosine kinase inhibitors: 3-substituted quinoline derivatives

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

(Imidazolylphenyl)pyrrol-2-one inhibitors of cardiac cAMP phosphodiesterase

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Olanzapine: a new typical antipsychotic drug

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Inhibition of hepatitis B surface antigen secretion on human hepatoma cells. Components from Rubia cordifolia

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis and biological characterization of 1,4,5,6-tetrahydropyrimidine and 2-amino-3,4,5,6-tetrahydropyridine derivatives as selective m1 agonists

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis and binding affinity of 2-phenylimidazo[1,2-alpha]pyridine derivatives for both central and peripheral benzodiazepine receptors. A new series of high-affinity and selective ligands for the peripheral type

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Regulation of Retinoidal Actions by Diazepinylbenzoic Acids.1Retinoid Synergists Which Activate the RXR−RAR Heterodimers

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Design, synthesis, and biological evaluation of conformationally constrained aci-reductone mimics of arachidonic acid

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Cell cycle arrest and antitumor activity of pironetin and its derivatives

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Tipranavir (PNU-140690): A Potent, Orally Bioavailable Nonpeptidic HIV Protease Inhibitor of the 5,6-Dihydro-4-hydroxy-2-pyrone Sulfonamide Class∇

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Hantzsch pyrrole synthesis on solid support

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Stereospecific synthesis, structure-activity relationship, and oral bioavailability of tetrahydropyrimidin-2-one HIV protease inhibitors

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Effect of tetrahydropyrimidine derivatives on protein-nucleic acids interaction. Type II restriction endonucleases as a model system

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Structural elements of the gamma-aminobutyric acid type A receptor conferring subtype selectivity for benzodiazepine site ligands

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Lamellarin alpha 20-sulfate, an inhibitor of HIV-1 integrase active against HIV-1 virus in cell culture

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Thiazolothiazepine inhibitors of HIV-1 integrase

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Total synthesis of ningalin B utilizing a heterocyclic azadiene Diels-Alder reaction and discovery of a new class of potent multidrug resistant (MDR) reversal agents

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Structure-activity studies on gossypol in tumor cell lines

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis and evaluation of quinoline carboxyguanidines as antidiabetic agents

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Selective small molecule inhibitors of glycogen synthase kinase-3 modulate glycogen metabolism and gene transcription

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Development of an efficient, regio- and stereoselective route to libraries based on the beta-D-glucose scaffold

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Guaiane dimers and germacranolide from Artemisia caruifolia

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Pyrazole ligands: structure-affinity/activity relationships and estrogen receptor-alpha-selective agonists.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

In vitro antiplasmodial activity of 4-phenylcoumarins from Exostema mexicanum

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis and antibacterial evaluation of certain quinolone derivatives

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

ATOP dyes. optimization of a multifunctional merocyanine chromophore for high refractive index modulation in photorefractive materials

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Oral gossypol in the treatment of patients with refractory metastatic breast cancer: a phase I/II clinical trial.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Catalytic functionalization of arenes and alkanes via C-H bond activation

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis of beta- and gamma-carbolines by the palladium-catalyzed iminoannulation of internal alkynes

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Montmorillonite KSF as an Inorganic, Water Stable, and Reusable Catalyst for the Knoevenagel Synthesis of Coumarin-3-carboxylic Acids

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Cyclic Dipeptides. 3.(1) Synthesis of Methyl (R)-6-[(tert-Butoxycarbonyl)amino]-4,5,6,7- tetrahydro-2-methyl-5-oxo-1,4-thiazepine-3-carboxylate and Its Hexahydro Analogues: Elaboration of a Novel Dual ACE/NEP Inhibitor

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Asymmetric Addition of Alkyllithium to Chiral Imines: alpha-Naphthylethyl Group as a Chiral Auxiliary

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

1,2-Diacetals: A New Opportunity for Organic Synthesis

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Palladium-catalyzed reactions of allenes

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Suzuki cross-coupling reactions of potassium alkenyltrifluoroborates

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Pd(II) acts simultaneously as a Lewis acid and as a transition-metal catalyst: synthesis of cyclic alkenyl ethers from acetylenic aldehydes

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Efficient synthesis of 3-furanosyl-6'-furanosylphosphinate through a tandem sequential radical process

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Transition Metal-Mediated Cycloaddition Reactions

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Domino Reactions in Organic Synthesis

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Carbeneminus signAlkyneminus signAlkene Cyclization Reactions

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Metal-Initiated Amination of Alkenes and Alkynes

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Bis(isoquinoline N-oxide) pincers as a new type of metal cation dual channel fluorosensor

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Total synthesis of cis-solamin

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Diastereoselective synthesis of the endo- and exo-spirotetronate subunits of the quartromicins. The first enantioselective Diels-Alder reaction of an acyclic (Z)-1,3-diene

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Antimicrobial activity of pyrrolizidine alkaloids from Heliotropium subulatum

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Novel approach for catalytic cyclopropanation of alkenes via (2-furyl)carbene complexes from 1-benzoyl-cis-1-buten-3-yne

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Rare-earth metal triflates in organic synthesis

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Phosphine-catalyzed annulation of thioamides and 2-alkynoates: a new synthesis of thiazolines

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Nucleophilic transition metal based cyclization of allenes

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Total synthesis and evaluation of lamellarin alpha 20-Sulfate analogues

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Olprinone: a phosphodiesterase III inhibitor with positive inotropic and vasodilator effects

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Bioactive 4-substituted-6-methyl-2-pyrones with promising cytotoxicity against A2780 and K562 cell lines

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Tandem reactions to construct heterocycles via phosphine-catalyzed umpolung addition and intramolecular conjugate addition

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis of beta- and gamma-carbolines by the palladium-catalyzed iminoannulation of alkynes

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Regioselective preparation of 2-substituted 3,4-diaryl pyrroles: a concise total synthesis of ningalin B

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Stereoselective synthesis of enynes by nickel-catalyzed cross-coupling of divinylic chalcogenides with alkynes

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis, structure-activity relationship, and evaluation of SR141716 analogues: development of central cannabinoid receptor ligands with lower lipophilicity.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Allosteric adenosine receptor modulation reduces hypersensitivity following peripheral inflammation by a central mechanism

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

The combinatorial synthesis of bicyclic privileged structures or privileged substructures.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

The catalytic hydroamination of alkynes

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis of spiro diphosphines and their application in asymmetric hydrogenation of ketones

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Reaction of enol ethers with alkynes catalyzed by transition metals: 5-exo-dig versus 6-endo-dig cyclizations via cyclopropyl platinum or gold carbene complexes

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

The rearrangement of 2,3-epoxysulfonates and its application to natural products syntheses: formal synthesis of (-)-aphanorphine and total syntheses of (-)-alpha-herbertenol and (-)-herbertenediol

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Early amidation approach to 3-[(4-amido)pyrrol-2-yl]-2-indolinones

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Catalytic asymmetric [3+2] cycloaddition of azomethine ylides. Development of a versatile stepwise, three-component reaction for diversity-oriented synthesis

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Construction of pyridine rings by metal-mediated [2 + 2 + 2] cycloaddition.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Glucose-lowering in a db/db mouse model by dihydropyridine diacid glycogen phosphorylase inhibitors

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Viridepyronone, a new antifungal 6-substituted 2H-pyran-2-one produced by Trichoderma viride

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Catalytic asymmetric sulfoxidation by chiral manganese complexes: acetylacetonate anions as chirality switches

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis and biological evaluation of 4-arylcoumarin analogues of combretastatins

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Optimization of the pharmacophore model for 5-HT7R antagonism. Design and synthesis of new naphtholactam and naphthosultam derivatives

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Syntheses, calcium channel agonist-antagonist modulation activities, and nitric oxide release studies of nitrooxyalkyl 1,4-dihydro-2,6-dimethyl-3-nitro-4-(2,1,3-benzoxadiazol-4-yl)pyridine-5-carboxylate racemates, enantiomers, and diastereomers

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Long-acting risperidone: a review of its use in schizophrenia

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

The effects of strontium ranelate on the risk of vertebral fracture in women with postmenopausal osteoporosis

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Cyanide-catalyzed cyclizations via aldimine coupling

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Oxidative C-C bond-forming reaction of electron-rich alkylbenzyl ether with trimethylvinyloxysilane

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Transition-metal-catalyzed reactions in heterocyclic synthesis

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis of oxygen- and nitrogen-containing heterocycles by ring-closing metathesis

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis of phosphorus and sulfur heterocycles via ring-closing olefin metathesis

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis of heterocycles via palladium pi-olefin and pi-alkyne chemistry

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Metalated heterocycles and their applications in synthetic organic chemistry

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Discovery of the first non-peptide full agonists for the human bradykinin B(2) receptor incorporating 4-(2-picolyloxy)quinoline and 1-(2-picolyl)benzimidazole frameworks

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

beta-Phenylethylamines and the isoquinoline alkaloids

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Comparison of fascaplysin and related alkaloids: a study of structures, cytotoxicities, and sources

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Transition-metal-catalyzed addition of heteroatom-hydrogen bonds to alkynes

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

2-pyrones possessing antimicrobial and cytotoxic activities

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

PtCl2-catalyzed cycloisomerizations of 5-en-1-yn-3-ol systems

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Substituted 3-imidazo[1,2-a]pyridin-3-yl- 4-(1,2,3,4-tetrahydro-[1,4]diazepino-[6,7,1-hi]indol-7-yl)pyrrole-2,5-diones as highly selective and potent inhibitors of glycogen synthase kinase-3.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Derivative of alpha,beta-dicyanostilbene: convenient precursor for the synthesis of diphenylmaleimide compounds, E-Z isomerization, crystal structure, and solid-state fluorescence

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Design, synthesis, and pharmacological evaluation of some 2-[4-morpholino]-3-aryl-5-substituted thiophenes as novel anti-inflammatory agents: generation of a novel anti-inflammatory pharmacophore

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Fluoride-Promoted Oxidation of Fischer Alkoxy Carbene Complexes: Stoichiometric and Catalytic Conditions

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Quantitative structure-activity relationship of sesquiterpene lactones as inhibitors of the transcription factor NF-kappaB

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Iron-catalyzed reactions in organic synthesis

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Gold(I)-catalyzed propargyl Claisen rearrangement

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Structure-activity relationship of 6-methylidene penems bearing tricyclic heterocycles as broad-spectrum beta-lactamase inhibitors: crystallographic structures show unexpected binding of 1,4-thiazepine intermediates

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Discovery of pyrano[3,4-b]indoles as potent and selective HCV NS5B polymerase inhibitors

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Catalytic transmetalation from group 6 Fischer carbene complexes: an emerging powerful tool in organic synthesis

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

The role of mitochondria for Ca2+ refilling of the endoplasmic reticulum

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis and antibacterial activities of 5-hydroxy-4-amino-2(5H)-furanones

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Identification of a novel cardenolide (2''-oxovoruscharin) from Calotropis procera and the hemisynthesis of novel derivatives displaying potent in vitro antitumor activities and high in vivo tolerance: structure-activity relationship analyses.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Cycloisomerization of 1,6-enynes using acetate as a nucleophile under palladium(II) catalysis

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Alpha-fluorinated ethers, thioethers, and amines: anomerically biased species.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Design, synthesis, biological evaluation and molecular docking of curcumin analogues as antioxidant, cyclooxygenase inhibitory and anti-inflammatory agents

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Reactions of vinyl acetate and vinyl trifluoroacetate with cationic diimine Pd(II) and Ni(II) alkyl complexes: identification of problems connected with copolymerizations of these monomers with ethylene

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Simple coumarins and analogues in medicinal chemistry: occurrence, synthesis and biological activity.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Secondary metabolites from endophytic Streptomyces aureofaciens CMUAc130 and their antifungal activity

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Risperidone: a review of its use in the treatment of bipolar mania

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis of coumarins, 4-hydroxycoumarins, and 4-hydroxyquinolinones by tellurium-triggered cyclizations.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Recent advances in transition metal catalyzed oxidation of organic substrates with molecular oxygen

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

2-Pyrone natural products and mimetics: isolation, characterisation and biological activity

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Some typical advances in the synthetic applications of allenes

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis and functionalization of indoles through palladium-catalyzed reactions

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Copper(II) acetate promoted intramolecular diamination of unactivated olefins

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis of spiro[4.5]trienones by intramolecular ipso-halocyclization of 4-(p-methoxyaryl)-1-alkynes

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Functionalized cyclobutenes via multicomponent thermal [2 + 2] cycloaddition reactions

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Chemistry. Palladium-catalyzed oxidation of organic chemicals with O2.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Palladium-catalyzed enantioselective conjugate addition of arylboronic acids

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Electrophilic activation of lactams with Tf2O and pyridine: expedient synthesis of (+/-)-tetraponerine T4

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Prevention of undesirable isomerization during olefin metathesis

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Application of olefin cross-metathesis to the synthesis of biologically active natural products

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

A selective turn-on fluorescent sensor for imaging copper in living cells.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Recent developments in isocyanide based multicomponent reactions in applied chemistry

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Pt(II)- or Au(III)-catalyzed [3+2] cycloaddition of metal-containing azomethine ylides: highly efficient synthesis of the mitosene skeleton

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

HIV integrase inhibitors with nucleobase scaffolds: discovery of a highly potent anti-HIV agent

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Hydrogen bond catalyzed direct reductive amination of ketones

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Investigation of the mechanism of action of 3-(4-bromophenyl)-5-acyloxymethyl-2,5-dihydrofuran-2-one against Candida albicans by flow cytometry

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

A pyrimidine-beta-carboline and other alkaloids from Annona foetida with antileishmanial activity

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Cortistatins A, B, C, and D, anti-angiogenic steroidal alkaloids, from the marine sponge Corticium simplex

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

A synthetic entry to furo[2,3-b]pyridin-4(1H)-ones and related furoquinolinones via iodocyclization

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Natural products in combinatorial chemistry: an andrographolide-based library

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Cancer cell mitochondria are direct proapoptotic targets for the marine antitumor drug lamellarin D.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

pi-Conjugated chelating polymers with charged iridium complexes in the backbones: synthesis, characterization, energy transfer, and electrochemical properties

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Ligand-modulated palladium-catalyzed aerobic alcohol oxidations

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

One-step assembly of carbamoyl-substituted heteroannelated [1,4]thiazepines

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Thermal Effects in the Organocatalytic Asymmetric Mannich Reaction

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Gold(I)-catalyzed stereoselective formation of functionalized 2,5-dihydrofurans

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Palladium(II)-catalyzed asymmetric synthesis of (Z)-alpha-alkylidene-gamma-butyrolactams from (Z)-N-allylic 2-Alkynamides. Total synthesis of (-)-isocynometrine

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis and characterization of palladium(II) and platinum(II) complexes with Schiff bases derivatives of 2-pyridincarboxyaldehyde. Study of their interaction with DNA.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Syntheses of polysubstituted furans: recent developments

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

beta-Phenylethylamines and the isoquinoline alkaloids

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

1,3-diketones from acid chlorides and ketones: a rapid and general one-pot synthesis of pyrazoles

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Interaction of 4-arylcoumarin analogues of combretastatins with microtubule network of HBL100 cells and binding to tubulin

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Series of new cationic iridium(III) complexes with tunable emission wavelength and excited state properties: structures, theoretical calculations, and photophysical and electrochemical properties

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Antimalarial 4-phenylcoumarins from the stem bark of Hintonia latiflora

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Kalanchosides A-C, new cytotoxic bufadienolides from the aerial parts of Kalanchoe gracilis

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Novel antitumor agent family of 1H-benzo[c,d]indol-2-one with flexible basic side chains: synthesis and biological evaluation

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Cationic palladium complex catalyzed highly enantioselective intramolecular addition of arylboronic acids to ketones. A convenient synthesis of optically active cycloalkanols

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Temporal mRNA profiles of inflammatory mediators in the murine 1-methyl-4-phenyl-1,2,3,6-tetrahydropyrimidine model of Parkinson's disease

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis of acyclic alpha,beta-unsaturated ketones via Pd(II)-catalyzed intermolecular reaction of alkynamides and alkenes

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

The Sonogashira reaction: a booming methodology in synthetic organic chemistry.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Hyrtinadine A, a bis-indole alkaloid from a marine sponge

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

A fascination with 1,2-diacetals.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Gold(I)-catalyzed oxidative rearrangements

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Two-faced reactivity of alkenes: cis- versus trans-aminopalladation in aerobic Pd-catalyzed intramolecular aza-Wacker reactions

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Asymmetric annulation toward pyrrolopiperazinones: concise enantioselective syntheses of pyrrole alkaloid natural products

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

3-Hydroxy-1,5-dihydro-pyrrol-2-one derivatives as advanced inhibitors of HIV integrase

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

The fascinating construction of pyridine ring systems by transition metal-catalysed [2 + 2 + 2] cycloaddition reactions

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Multi-component syntheses of heterocycles by transition-metal catalysis

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Intramolecular aminopalladation of alkenes as a key step to pyrrolidines and related heterocycles

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Heterocycle synthesis by copper facilitated addition of heteroatoms to alkenes, alkynes and arenes

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Cationic Pd(II)-catalyzed enantioselective cyclization of aroylmethyl 2-alkynoates initiated by carbopalladation of alkynes with arylboronic acids

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Gold-catalyzed organic reactions

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Cu-Catalyzed Tandem C−N Bond Formation for the Synthesis of Pyrroles and Heteroarylpyrroles

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Ultrasonic-promoted three-component synthesis of some biologically active 1,2,5,6-tetrahydropyrimidines

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Systemic fungicidal activity of 1,4-oxathiin derivatives

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Pyrido[1,2-a]pyrimidin-4-one Derivatives as a Novel Class of Selective Aldose Reductase Inhibitors Exhibiting Antioxidant Activity

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Sequential Cu-catalyzed amidation-base-mediated camps cyclization: a two-step synthesis of 2-Aryl-4-quinolones from o-halophenones

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Recent progress in the pharmacology of imidazo[1,2-a]pyridines

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Flexible synthetic routes to poison-frog alkaloids of the 5,8-disubstituted indolizidine-class I: synthesis of common lactam chiral building blocks and application to the synthesis of (-)-203A, (-)-205A, and (-)-219F.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

BODIPY dyes and their derivatives: syntheses and spectroscopic properties.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Role of environmental toxins in endemic (Balkan) nephropathy. October 2006, Zagreb, Croatia

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

C-C, C-O, C-N bond formation on sp2 carbon by Pd(II)-catalyzed reactions involving oxidant agents

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Sequential rhodium-catalyzed stereo- and regioselective addition of organoboron derivatives to the alkyl 4-hydroxy-2-alkynoates/lactonizaction reaction.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Antitumor activity of 4-arylcoumarins from endophytic Streptomyces aureofaciens CMUAc130.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Lamellarins and related pyrrole-derived alkaloids from marine organisms

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis of multisubstituted 2-(dihydrofuran-2(3H)-ylidene)acetates via intramolecular carboalkoxylation by platinum-olefin catalyst system

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

High mobility single-crystal field-effect transistors from bisindoloquinoline semiconductors

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Total synthesis of the indolizidine alkaloid tashiromine

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Selective synthesis of spiro[4,5]trienyl acetates via an intramolecular electrophilic ipso-iodocyclization process

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Preparation and intramolecular [2+2]-photocycloaddition of 1,5-dihydropyrrol-2-ones and 5,6-dihydro-1H-pyridin-2-ones with C-, N-, and O-linked alkenyl side chains at the 4-position

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Intermolecular Radical Addition of Alkylthio- and Arylthiodiphenylphosphines to Terminal Alkynes

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Tetramic and tetronic acids: an update on new derivatives and biological aspects

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

ent-Labdane diterpenoid lactone stereoisomers from Andrographis paniculata

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Ring-closing metathesis: novel routes to aromatic heterocycles

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

A mild, one-pot synthesis of 4-quinolones via sequential Pd-catalyzed amidation and base-promoted cyclization

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Design, synthesis, and biological evaluation of novel 3-aryl-4-(1H-indole-3yl)-1,5-dihydro-2H-pyrrole-2-ones as vascular endothelial growth factor receptor (VEGF-R) inhibitors

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Rhodium-catalyzed highly enantio- and diastereoselective cotrimerization of alkenes and dialkyl acetylenedicarboxylates leading to furylcyclopropanes

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Coinage metal-assisted synthesis of heterocycles.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Gold-Catalyzed Organic Transformations

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Ag-mediated reactions: coupling and heterocyclization reactions

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

The conformational rigidity of butane-1,2-diacetals as a powerful synthetic tool

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Amino(oligo)thiophene-based environmentally sensitive biomembrane chromophores

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Cu-catalyzed azide-alkyne cycloaddition

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Copper-mediated coupling reactions and their applications in natural products and designed biomolecules synthesis

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Design of a highly efficient and water-tolerant sulfonic acid nanoreactor based on tunable ordered porous silica for the von Pechmann reaction

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Au-containing all-carbon 1,3-dipoles: generation and [3+2] cycloaddition reactions

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Small molecule modulators of toll-like receptors

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Et3N-induced demethylation-annulation of 3-alkynyl-4-methoxy-2-pyridones and structurally related compounds in the synthesis of furan-fused heterocycles

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

The Chemistry of 4-Hydroxyquinolines

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Strategies for the total synthesis of C2-C11 cyclized cembranoids

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Development, scope and mechanisms of multicomponent reactions of asymmetric electron-deficient alkynes with amines and formaldehyde

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Oligosubstituted pyrroles directly from substituted methyl isocyanides and acetylenes

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Analyte-triggered gelation: initiating self-assembly via oxidation-induced planarization

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Solid-phase synthesis of biologically active benzoannelated nitrogen heterocycles: an update.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis of 4-arylcoumarins via Cu-catalyzed hydroarylation with arylboronic acids

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Regio- and chemoselective synthesis of fully substituted thiophenes

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Nanoparticle-supported and magnetically recoverable ruthenium hydroxide catalyst: efficient hydration of nitriles to amides in aqueous medium

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Biomimetic synthesis toward the transtaganolides/basiliolides

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthetic medicinal chemistry of selected antimalarial natural products

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Highly enantioselective hydrogenation of enamides catalyzed by chiral phosphoric acids

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Functional Oligothiophenes: Molecular Design for Multidimensional Nanoarchitectures and Their Applications†

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

An efficient synthesis of 2,5-dihydrofuran-fused bicyclic skeletons via the Pd(II)-catalyzed tandem-cyclization reaction of 1,omega-bisallenols

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Direct amination of azoles via catalytic C-H, N-H coupling

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Copper-catalyzed domino rearrangement/dehydrogenation oxidation/carbene oxidation for one-pot regiospecific synthesis of highly functionalized polysubstituted furans

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Recent advances in the synthesis of indole and quinoline derivatives through cascade reactions.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Recent advances in the Friedländer reaction

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Copper(0)-induced deselenative insertion of N,N-disubstituted selenoamides into acetylenic C-H bond leading to propargylamines

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Construction of nitrogen-containing heterocycles by C-H bond functionalization

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Solvent-free heterocyclic synthesis

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Discovery of a new class of protein farnesyltransferase inhibitors in the arylthiophene series

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Single-electron transfer and single-electron transfer degenerative chain transfer living radical polymerization

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Escape from flatland: increasing saturation as an approach to improving clinical success

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Stereoselective synthesis of (E)-2-en-4-ynoic acids with ynolates: catalytic conversion to tetronic acids and 2-pyrones

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Perylenequinone natural products: total synthesis of hypocrellin A.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Control of chemoselectivity by counteranions of cationic palladium complexes: a convenient enantioselective synthesis of dihydrocoumarins

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

One-pot silver-catalyzed and PIDa-mediated sequential reactions: synthesis of polysubstituted pyrroles directly from alkynoates and amines

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthetic approach to polysubstituted furans: an efficient addition/oxidative cyclization of alkynoates and 1,3-dicarbonyl compounds

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

A new catalyst for organic synthesis: mercuric triflate

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Functionalization of organic molecules by transition-metal-catalyzed C(sp3)-H activation

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Inhibition of mitochondrial respiration mediates apoptosis induced by the anti-tumoral alkaloid lamellarin D.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Dihydrobenzo[1,4]oxathiine: A multi-potent pharmacophoric heterocyclic nucleus.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Gold-catalyzed intermolecular hydrophenoxylation of unactivated internal alkynes

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

The discovery and structure-activity relationships of pyrano[3,4-b]indole based inhibitors of hepatitis C virus NS5B polymerase

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis and biological evaluation of some thio containing pyrrolo [2,3-d]pyrimidine derivatives for their anti-inflammatory and anti-microbial activities

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis of beta- and gamma-carbolinones via Pd-catalyzed direct dehydrogenative annulation (DDA) of indole-carboxamides with alkynes using air as the oxidant.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Copper-catalyzed intramolecular C-H oxidation/acylation of formyl-N-arylformamides leading to indoline-2,3-diones

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis and structure-activity relationship of 6-arylureido-3-pyrrol-2-ylmethylideneindolin-2-one derivatives as potent receptor tyrosine kinase inhibitors

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Cu (I)-catalyzed synthesis of polysubstituted pyrroles from dialkyl ethylenedicarboxylates and beta-enamino ketones or esters in the presence of O2

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Nano-Cu(2)O-catalyzed formation of C-C and C-O bonds: one-pot domino process for regioselective synthesis of α-carbonyl Furans from electron-deficient alkynes and 2-yn-1-ols

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Multicomponent reactions for the synthesis of pyrroles.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Isocyanoacetate derivatives: synthesis, reactivity, and application.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Recent advances in transition metal-catalyzed N-atom transfer reactions of azides

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis, selective anti-Helicobacter pylori activity, and cytotoxicity of novel N-substituted-2-oxo-2H-1-benzopyran-3-carboxamides

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Supramolecular Assemblies in Ionic Liquid Catalysis for Aza-Michael Reaction

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Cooperative Catalysis with Metal and Secondary Amine: Synthesis of 2-Substituted Quinolines via Addition/Cycloisomerization Cascade

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Design, synthesis, and preclinical evaluation of new 5,6- (or 6,7-) disubstituted-2-(fluorophenyl)quinolin-4-one derivatives as potent antitumor agents.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Cu(I)−Amido Complexes in the Ullmann Reaction: Reactions of Cu(I)−Amido Complexes with Iodoarenes with and without Autocatalysis by CuI

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

3-Arylisoquinolines as novel topoisomerase I inhibitors

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

An atom-economic synthesis of nitrogen heterocycles from alkynes

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Total synthesis of lamellarins D, H, and R and ningalin B.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Efficacy of antidepressants and benzodiazepines in minor depression: systematic review and meta-analysis

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Enhanced functionality for donor-acceptor oligothiophenes by means of inclusion of BODIPY: synthesis, electrochemistry, photophysics, and model chemistry.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis and NLO properties of new trans 2-(thiophen-2-yl)vinyl heteroaromatic iodides.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Gold-catalyzed nucleophilic cyclization of functionalized allenes: a powerful access to carbo- and heterocycles

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Vipirinin, a coumarin-based HIV-1 Vpr inhibitor, interacts with a hydrophobic region of VPR.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Discovery and synthesis of novel 3-phenylcoumarin derivatives as antidepressant agents

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Gold-Catalyzed Carbon−Heteroatom Bond-Forming Reactions

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Development of methods for the synthesis of libraries of substituted maleimides and α,β-unsaturated-γ-butyrolactams

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Antifungal, cytotoxic and SAR studies of a series of N-alkyl, N-aryl and N-alkylphenyl-1,4-pyrrolediones and related compounds

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

"One-pot" multicomponent approach to indolizines and pyrido[1,2-a]indoles

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Use of nonfunctionalized enamides and enecarbamates in asymmetric synthesis

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Phosphine-catalyzed [3+2] annulations of γ-functionalized butynoates and 1C,3O-bisnucleophiles: highly selective reagent-controlled pathways to polysubstituted furans.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Perspectives on the structural and biosynthetic interrelationships between oxygenated furanocembranoids and their polycyclic congeners found in corals

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Gold(III) chloride catalyzed regioselective synthesis of pyrano[3,4-b]indol-1(9H)-ones and evaluation of anticancer potential towards human cervix adenocarcinoma

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Copper-catalyzed aerobic oxidative intramolecular alkene C-H amination leading to N-heterocycles

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Study on the anticancer activity of coumarin derivatives by molecular modeling.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

A facile synthesis of highly functionalized 4-arylcoumarins via Kostanecki reactions mediated by DBU.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Advances in the chemistry of tetrahydroquinolines.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

One-pot two-component [3 + 2] cycloaddition/annulation protocol for the synthesis of highly functionalized thiophene derivatives

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Copper-catalyzed coupling of oxime acetates with aldehydes: a new strategy for synthesis of pyridines

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Convenient Synthesis of 3-Vinyl and 3-Styryl Coumarins

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Recent progress in synthesis and bioactivity studies of indolizines

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Identification of pyrido[1,2-α]pyrimidine-4-ones as new molecules improving the transcriptional functions of estrogen-related receptor α.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Photoswitchable organic mixed valence in dithienylcyclopentene systems with tertiary amine redox centers

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Organic Dyes Containing a Coplanar Indacenodithiophene Bridge for High-Performance Dye-Sensitized Solar Cells

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Phase separation as a strategy toward controlling dilution effects in macrocyclic Glaser-Hay couplings

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis and in vitro anticancer activity of 6,7-methylenedioxy (or 5-hydroxy-6-methoxy)-2-(substituted selenophenyl)quinolin-4-one analogs

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

1,2-Benzothiazine 1,1-dioxide carboxylate derivatives as novel potent inhibitors of aldose reductase

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Mechanisms of nucleophilic organocopper(I) reactions.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

The Prins reaction using ketones: rationalization and application toward the synthesis of the portentol skeleton

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Silver-Mediated C–H Activation: Oxidative Coupling/Cyclization of N-Arylimines and Alkynes for the Synthesis of Quinolines

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Rhodium catalyzed chelation-assisted C-H bond functionalization reactions

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Antioxidant properties of 4-quinolones and structurally related flavones

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Evidence for alkene cis-aminocupration, an aminooxygenation case study: kinetics, EPR spectroscopy, and DFT calculations

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Gold-catalyzed furan/yne cyclizations for the regiodefined assembly of multisubstituted protected 1-naphthols

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

4-Aryl-2-quinolones from 3,3-diarylacrylamides through intramolecular copper-catalyzed C-H functionalization/C-N bond formation

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Recent advances in transition-metal catalyzed reactions using molecular oxygen as the oxidant.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Intramolecular ipso-halocyclization of 4-(p-unsubstituted-aryl)-1-alkynes leading to spiro[4,5]trienones: scope, application, and mechanistic investigations

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Palladium-catalyzed intramolecular hydroarylation of 4-benzofuranyl alkynoates. Approach to angelicin derivatives

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

C-C, C-O and C-N bond formation via rhodium(III)-catalyzed oxidative C-H activation.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

7-Ethynylcoumarins: selective inhibitors of human cytochrome P450s 1A1 and 1A2.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Chemistry and biology of fascaplysin, a potent marine-derived CDK-4 inhibitor

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Recent developments and biological activities of thiazolidinone derivatives: a review.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Hydroxyl-directed ruthenium-catalyzed C-H bond functionalization: versatile access to fluorescent pyrans

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Phosphine/palladium-catalyzed syntheses of alkylidene phthalans, 3-deoxyisoochracinic acid, isoochracinic acid, and isoochracinol

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Naphthalenones from a Perenniporia sp. inhabiting the larva of a phytophagous weevil, Euops chinesis

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

From biomass to medicines. A simple synthesis of indolo[3,2-c]quinolines, antimalarial alkaloid isocryptolepine, and its derivatives

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Palladium-catalyzed oxidation of unsaturated hydrocarbons using molecular oxygen

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Copper(II)/iron(III) co-catalyzed intermolecular diamination of alkynes: facile synthesis of imidazopyridines.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis of imidazopyridines from the Morita-Baylis-Hillman acetates of nitroalkenes and convenient access to Alpidem and Zolpidem

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Completely OH-selective FeCl3-catalyzed Prins cyclization: highly stereoselective synthesis of 4-OH-tetrahydropyrans

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Design, synthesis, and pharmacological characterization of N- and O-substituted 5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]azepin-3-ol analogues: novel 5-HT(2A)/5-HT(2C) receptor agonists with pro-cognitive properties

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Transition metal-mediated synthesis of monocyclic aromatic heterocycles

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis of isocoumarin derivatives by copper-catalyzed addition of o-halobenzoic acids to active internal alkynes

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Arylglyoxals in synthesis of heterocyclic compounds

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Carboxylate-assisted ruthenium-catalyzed alkyne annulations by C-H/Het-H bond functionalizations

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Efficacy of cytisine in helping smokers quit: systematic review and meta-analysis

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Copper-catalyzed C-O bond formation: an efficient one-pot highly regioselective synthesis of furans from (2-furyl)carbene complexes.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Development of four-component synthesis of tetra- and pentasubstituted polyfunctional dihydropyrroles: free permutation and combination of aromatic and aliphatic amines

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Modular pyridine synthesis from oximes and enals through synergistic copper/iminium catalysis.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Current developments of coumarin compounds in medicinal chemistry.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Atropisomers of arylmaleimides: stereodynamics and absolute configuration

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Thiophene-core estrogen receptor ligands having superagonist activity.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Triazolothiadiazoles and triazolothiadiazines--biologically attractive scaffolds

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Overcoming product inhibition in catalysis of the intramolecular Schmidt reaction

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Copper-catalyzed direct synthesis of iodoenamides from ketoximes

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Aerobic copper-catalyzed organic reactions

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Bioactive compounds from the roots of Strophioblachia fimbricalyx.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Coumarin derivatives protect against ischemic brain injury in rats

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

TEMPO-catalyzed aerobic oxygenation and nitrogenation of olefins via C═C double-bond cleavage

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Chemicals from Coal Coking

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Iron-catalyzed ring-opening azidation and allylation of O-heterocycles

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Silver-mediated oxidative C-H/P-H functionalization: an efficient route for the synthesis of benzo[b]phosphole oxides.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

CuI-catalyzed aerobic oxidative α-aminaton cyclization of ketones to access aryl or alkenyl-substituted imidazoheterocycles

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

4-Trifluoromethyl-substituted coumarins with large Stokes shifts: synthesis, bioconjugates, and their use in super-resolution fluorescence microscopy

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Flexible routes to thiophenes

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Palladium-catalyzed coupling of alkynes with unactivated alkenes in ionic liquids: a regio- and stereoselective synthesis of functionalized 1,6-dienes and their analogues.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

6-Phosphorylated phenanthridines from 2-isocyanobiphenyls via radical C-P and C-C bond formation.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Pyrrolizines: Promising scaffolds for anticancer drugs

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

DDQ-mediated oxidative coupling: an approach to 2,3-dicyanofuran (thiophene).

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

A new prenylated indole derivative from endophytic actinobacteria Streptomyces sp. neau-D50.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Potent and Selective Double-Headed Thiophene-2-carboximidamide Inhibitors of Neuronal Nitric Oxide Synthase for the Treatment of Melanoma

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Copper-promoted oxidative coupling of enamides and alkynes for the synthesis of substituted pyrroles

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Design, synthesis and pharmacological evaluation of novel pyrrolizine derivatives as potential anticancer agents

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Biosynthetic potential-based strain prioritization for natural product discovery: a showcase for diterpenoid-producing actinomycetes

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Total Synthesis of (±)-Distomadines A and B

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Recent advances in the structural library of functionalized quinazoline and quinazolinone scaffolds: synthetic approaches and multifarious applications.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Pd-catalyzed branching cyclizations of enediyne-imides toward furo[2,3-b]pyridines

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis, crystal structure and biological evaluation of some novel 1,2,4-triazolo[3,4-b]-1,3,4-thiadiazoles and 1,2,4-triazolo[3,4-b]-1,3,4-thiadiazines.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Copper(II)-catalyzed carbon-carbon triple bond cleavage of internal alkynes for the synthesis of annulated indolizines

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Copper-mediated oxidative transformation of N-allyl enamine carboxylates toward synthesis of azaheterocycles

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis of β-allylbutenolides via one-pot copper-catalyzed hydroallylation/cyclization of γ-hydroxybutynoate derivatives

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Optimization of small-molecule inhibitors of influenza virus polymerase: from thiophene-3-carboxamide to polyamido scaffolds

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Phthalides and phthalans: synthetic methodologies and their applications in the total synthesis.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Total synthesis of the antitumor natural product polycarcin V and evaluation of its DNA binding profile

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

4-Quinolone-3-carboxylic acids as cell-permeable inhibitors of protein tyrosine phosphatase 1B.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Silver-catalyzed synthesis of 3-phosphorated coumarins via radical cyclization of alkynoates and dialkyl H-phosphonates.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Diarylrhodates as promising active catalysts for the arylation of vinyl ethers with Grignard reagents.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis and structure-activity relationships of lapacho analogues. 2. Modification of the basic naphtho[2,3-b]furan-4,9-dione, redox activation, and suppression of human keratinocyte hyperproliferation by 8-hydroxynaphtho[2,3-b]thiophene-4,9-dione

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Copper-catalyzed annulation of heteroaromatic β-halo-α,β-unsaturated carboxylic acids with alkynes for the synthesis of indolo[2,3-c]pyrane-1-ones and thieno[2,3-c]pyrane-7-ones

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Copper(I)-catalyzed multicomponent reaction providing a new access to fully substituted thiophene derivatives

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Ralfuranone Is Produced by an Alternative Aryl-Substituted γ-Lactone Biosynthetic Route in Ralstonia solanacearum

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

A broadly applicable and practical oligomeric (salen) Co catalyst for enantioselective epoxide ring-opening reactions

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Copper-catalyzed direct trifluoromethylation of propiolates: construction of trifluoromethylated coumarins.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Rh(III)-catalyzed cyclopropanation initiated by C-H activation: ligand development enables a diastereoselective [2 + 1] annulation of N-enoxyphthalimides and alkenes

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Multicomponent [5 + 2] cycloaddition reaction for the synthesis of 1,4-diazepines: isolation and reactivity of azomethine ylides

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthetic methods for compounds having CF3-S units on carbon by trifluoromethylation, trifluoromethylthiolation, triflylation, and related reactions

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis and cytotoxicity of thieno[2,3-b]pyridine and furo[2,3-b]pyridine derivatives

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Direct synthesis of polysubstituted 2-aminothiophenes by Cu(II)-catalyzed addition/oxidative cyclization of alkynoates with thioamides

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Unexpected regioselective carbon-hydrogen bond activation/cyclization of indolyl aldehydes or ketones with alkynes to benzo-fused oxindoles

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Analysis of the structural diversity, substitution patterns, and frequency of nitrogen heterocycles among U.S. FDA approved pharmaceuticals

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Active compounds from a diverse library of triazolothiadiazole and triazolothiadiazine scaffolds: synthesis, crystal structure determination, cytotoxicity, cholinesterase inhibitory activity, and binding mode analysis

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Iron(III) chloride and diorganyl diselenides-mediated 6-endo-dig cyclization of arylpropiolates and arylpropiolamides leading to 3-organoselenyl-2H-coumarins and 3-organoselenyl-quinolinones

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Ligand-controlled regiodivergent pathways of rhodium(III)-catalyzed dihydroisoquinolone synthesis: experimental and computational studies of different cyclopentadienyl ligands.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Medicinal chemistry optimization of antiplasmodial imidazopyridazine hits from high throughput screening of a softfocus kinase library: part 2.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Biased multicomponent reactions to develop novel bromodomain inhibitors.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Gold-catalyzed dearomative spirocyclization of aryl alkynoate esters

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Copper-catalyzed regioselective synthesis of furan via tandem cycloaddition of ketone with an unsaturated carboxylic acid under air.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Lead optimization and modulation of hERG activity in a series of aminooxazoline xanthene β-site amyloid precursor protein cleaving enzyme (BACE1) inhibitors

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Chemistry of α-oxoesters: a powerful tool for the synthesis of heterocycles.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthetic approaches, functionalization and therapeutic potential of quinazoline and quinazolinone skeletons: the advances continue.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Sequential One-Pot Synthesis of Tri- and Tetrasubstituted Thiophenes and Fluorescent Push-Pull Thiophene Acrylates Involving (Het)aryl Dithioesters as Thiocarbonyl Precursors

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Preparation of 3-Acyl-4-arylcoumarins via Metal-Free Tandem Oxidative Acylation/Cyclization between Alkynoates with Aldehydes.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

C–H Arylation of Unsubstituted Furan and Thiophene with Acceptor Bromides: Access to Donor–Acceptor–Donor-Type Building Blocks for Organic Electronics

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Silver-mediated radical cyclization of alkynoates and α-keto acids leading to coumarins via cascade double C-C bond formation

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Nickel-catalyzed alkynylation of anisoles via C-O bond cleavage

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Regioselective palladium-catalyzed decarboxylative cross-coupling reaction of alkenyl acids with coumarins: synthesis of 3-styrylcoumarin compounds.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Design and optimization of a series of 1-sulfonylpyrazolo[4,3-b]pyridines as selective c-Met inhibitors.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Bi(OTf)3-mediated cycloisomerization of γ-alkynyl arylketones: application to the synthesis of substituted furans

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Three-component domino process for the pyrrolizine skeleton via [3 + 2]-cycloaddition-enamine cyclization triggered by a gold catalyst

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Visible-light-mediated radical aryldifluoroacetylation of alkynes with ethyl bromodifluoroacetate for the synthesis of 3-difluoroacetylated coumarins.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Substrate activation strategies in rhodium(III)-catalyzed selective functionalization of arenes

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Thiazolidine-2,4-dione derivatives: programmed chemical weapons for key protein targets of various pathological conditions

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Divergent synthesis of 4,6-diarylated pyridin-2(1H)-ones from chalcones: novel access to 2,4,6-triaryl pyridines

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Application of Thio-Ugi Adducts for the Preparation of Benzo[b]thiophene and S-Heterocycle Library via Copper Catalyzed Intramolecular C-S Bond Formation.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Chiral Phosphoric Acid Catalyzed Asymmetric Synthesis of 2-Substituted 2,3-Dihydro-4-quinolones by a Protecting-Group-Free Approach

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Coumarin heterocyclic derivatives: chemical synthesis and biological activity

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Expedient Access to 2,3-Dihydropyridines from Unsaturated Oximes by Rh(III)-Catalyzed C-H Activation

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Copper(I)-Catalyzed Radical Addition of Acetophenones to Alkynes in Furan Synthesis

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Copper-Catalyzed Diazo Cross-/Homo-Coupling toward Tetrasubstituted Olefins and Applications on the Synthesis of Maleimide Derivatives.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Deformylative Intramolecular Hydroarylation: Synthesis of Benzo[e]pyrido[1,2-a]indoles

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Novel 2H-chromen-2-one derivatives of resveratrol: Design, synthesis, modeling and use as human monoamine oxidase inhibitors

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Transition-Metal-Catalyzed Cleavage of C-N Single Bonds

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Phenyliodine(III) Diacetate Mediated Oxidative Cyclization of 1-Alkenoyl-1-carbamoyl Cycloalkanes: Access to Spiro-Fused Dihydrofuran-3(2H)-ones

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Copper(II)-Mediated Aerobic Synthesis of Imidazo[1,2-a]pyridines via Cascade Aminomethylation/Cycloisomerization of Alkynes

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Rhodium-catalysed syn-carboamination of alkenes via a transient directing group

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

LDA-Promoted Synthesis of 3-Amino Furans by Selective Lithiation of Enaminones

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Nickel-Catalyzed Formal Homocoupling of Methoxyarenes for the Synthesis of Symmetrical Biaryls via C-O Bond Cleavage.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Pyrrolo-[3,2-b]pyrroles for Photochromic Analysis of Halocarbons.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Manganese- and Borane-Mediated Synthesis of Isobenzofuranones from Aromatic Esters and Oxiranes via C-H Bond Activation

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Continuous Flow Magnesiation or Zincation of Acrylonitriles, Acrylates, and Nitroolefins. Application to the Synthesis of Butenolides

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Geranylated 4-Phenylcoumarins Exhibit Anticancer Effects against Human Prostate Cancer Cells through Caspase-Independent Mechanism

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Quinazolines and quinazolinones as ubiquitous structural fragments in medicinal chemistry: An update on the development of synthetic methods and pharmacological diversification.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Isocoumarins, miraculous natural products blessed with diverse pharmacological activities.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Copper-Mediated [3 + 2] Oxidative Cyclization Reaction of N-Tosylhydrazones and β-Ketoesters: Synthesis of 2,3,5-Trisubstituted Furans.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Rhodium(III)-Catalyzed Tandem [2+2+2] Annulation-Lactamization of Anilides with Two Alkynoates via Cleavage of Two Adjacent C-H or C-H/C-O bonds.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Visible-Light-Promoted Dual C-C Bond Formations of Alkynoates via a Domino Radical Addition/Cyclization Reaction: A Synthesis of Coumarins

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Pd(II)-Catalyzed Tandem Heterocyclization of 1-(1-Alkynyl)cyclopropyl Oxime Derivatives for the Synthesis of Functionalized Pyrroles

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Charting the Chemical Reactivity Space of 2,3-Substituted Furo[2,3-b]pyridines Synthesized via the Heterocyclization of Pyridine-N-oxide Derivatives

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Coumarin-thiazole and -oxadiazole derivatives: Synthesis, bioactivity and docking studies for aldose/aldehyde reductase inhibitors

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Direct Tryptophols Synthesis from 2-Vinylanilines and Alkynes via C≡C Triple Bond Cleavage and Dioxygen Activation.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis of trifluoromethylthiolated pyridinones through the copper-mediated trifluoromethylthiolation of iodopyridinones

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

De novo protecting-group-free total synthesis of (+)-muricadienin, (+)-ancepsenolide and (+)-3-hexadecyl-5-methylfuran-2(5H)-one

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Regiocontrolled Coupling of Aromatic and Vinylic Amides with α-Allenols To Form γ-Lactams via Rhodium(III)-Catalyzed C-H Activation

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Sulfoximines from a Medicinal Chemist's Perspective: Physicochemical and in vitro Parameters Relevant for Drug Discovery

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Symmetrical aryl linked bis-iminothiazolidinones as new chemical entities for the inhibition of monoamine oxidases: Synthesis, in vitro biological evaluation and molecular modelling analysis.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Assembly of Polysubstituted Maleimides via Palladium-Catalyzed Cyclization Reaction of Alkynes with Isocyanides

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Transition Metal-Catalyzed C-H Amination: Scope, Mechanism, and Applications.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Oxidative C-H/C-H Coupling Reactions between Two (Hetero)arenes

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Visible-Light-Induced C2 Alkylation of Pyridine N-Oxides.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Novel Pieces for the Emerging Picture of Sulfoximines in Drug Discovery: Synthesis and Evaluation of Sulfoximine Analogues of Marketed Drugs and Advanced Clinical Candidates

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Manganese(I)-Catalyzed Dispersion-Enabled C-H/C-C Activation

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

1,2-Benzothiazines from Sulfoximines and Allyl Methyl Carbonate by Rhodium-Catalyzed Cross-Coupling and Oxidative Cyclization

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Manganese-catalyzed allylation via sequential C-H and C-C/C-Het bond activation.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Quinolinic carboxylic acid derivatives as potential multi-target compounds for neurodegeneration: monoamine oxidase and cholinesterase inhibition

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Unusual Blue-Shifted Acid-Responsive Photoluminescence Behavior in 6-Amino-8-cyanobenzo[1,2-b]indolizines

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Catalytic Asymmetric Synthesis of Butenolides and Butyrolactones

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Preparation of 3-Iodoquinolines from N-Tosyl-2-propynylamines with Diaryliodonium Triflate and N-Iodosuccinimide.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Exploration of aroyl/heteroaroyl iminothiazolines featuring 2,4,5-trichlorophenyl moiety as a new class of potent, selective, and in vitro efficacious glucosidase inhibitors.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Iron-Catalyzed Intermolecular Hydrothiolation of Internal Alkynes with Thiosalicylic Acids, and Sequential Intramolecular Cyclization Reaction

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Rhodium(III)-Catalyzed Synthesis of Naphthols via C-H Activation of Sulfoxonium Ylides

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

The Tetraarylpyrrolo[3,2-b]pyrroles-From Serendipitous Discovery to Promising Heterocyclic Optoelectronic Materials

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Direct Synthesis of 4-Quinolones via Copper-Catalyzed Anilines and Alkynes.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Exploration of thioxothiazolidinone-sulfonate conjugates as a new class of aldehyde/aldose reductase inhibitors: A synthetic and computational investigation

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

A Direct Cycloaminative Approach to Imidazole Derivatives via Dual C-H Functionalization.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Enantio- and Diastereoselective Betti/aza-Michael Sequence: Single Operated Preparation of Chiral 1,3-Disubstituted Isoindolines.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis of Functionalized Pyridines via Cu(II)-Catalyzed One-Pot Cascade Reactions of Inactivated Saturated Ketones with Electron-Deficient Enamines.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Visible-light-mediated direct difluoromethylation of alkynoates: synthesis of 3-difluoromethylated coumarins

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Aromatic C-H addition of ketones to imines enabled by manganese catalysis

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Copper-Catalyzed Oxidative Cyclization of Maleimides with Amines and Alkyne Esters: Direct Access to Fully Substituted Dihydropyrroles and Pyrrole Derivatives

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Iron-Catalyzed Indolizine Synthesis from Pyridines, Diazo Compounds, and Alkynes.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

From Ketones, Amines, and Carbon Monoxide to 4-Quinolones: Palladium-Catalyzed Oxidative Carbonylation.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Recent advance in oxazole-based medicinal chemistry

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Ruthenium-Catalyzed Hydrogenation of Carbocyclic Aromatic Amines: Access to Chiral Exocyclic Amines

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

A new entry into the portfolio of α-glucosidase inhibitors as potent therapeutics for type 2 diabetes: Design, bioevaluation and one-pot multi-component synthesis of diamine-bridged coumarinyl oxadiazole conjugates.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Inert C-H Bond Transformations Enabled by Organometallic Manganese Catalysis.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Divergent Synthesis of Quinolones and Dihydroepindolidiones via Cu(I)-Catalyzed Cyclization of Anilines with Alkynes

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

A lesson for site-selective C-H functionalization on 2-pyridones: radical, organometallic, directing group and steric controls.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Copper-Catalyzed Oxygenation Approach to Oxazoles from Amines, Alkynes, and Molecular Oxygen.

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Photoredox-Catalyzed Cascade Radical Cyclization of Ester Arylpropiolates with CF3SO2Cl To Construct 3-Trifluoromethyl Coumarin Derivatives

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Developing hybrid molecule therapeutics for diverse enzyme inhibitory action: Active role of coumarin-based structural leads in drug discovery

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

PIDA/I2-Mediated α- and β-C(sp3)-H Bond Dual Functionalization of Tertiary Amines

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Palladium-catalyzed cascade carboesterification of norbornene with alkynes

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Visible-light-promoted radical acylation/cyclization of alkynoates with aldehydes for the synthesis of 3-acylcoumarins

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

One-pot four-component synthesis of thiazolidin-2-imines using CuI/ZnII dual catalysis: A new class of acetylcholinesterase inhibitors

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Ru-Catalyzed Regioselective Cascade Annulation of Acrylamides with 2-Alkynoates for the Synthesis of Various 6-Oxo Nicotinic Acid Esters

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Indium-Catalyzed Denitrogenative Transannulation of Pyridotriazoles: Synthesis of Pyrido[1,2- a]indoles

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Progress in the Chemistry of Tetrahydroquinolines

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Probing the high potency of pyrazolyl pyrimidinetriones and thioxopyrimidinediones as selective and efficient non-nucleotide inhibitors of recombinant human ectonucleotidases

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Nickel-catalyzed oxidative C-H/N-H annulation of -heteroaromatic compounds with alkynes

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

An efficient light on-off one-pot method for the synthesis of 3-styryl coumarins from aryl alkynoates

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Rh(III)-Catalyzed Oxidative Annulation of Sulfoximines with Arylalkynyl Silanes via Desilylation

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis of Furanone-Fused 1,2-Benzothiazine by Rh(III)-Catalyzed C-H Activation: Regioselective Oxidative Annulation Leading to in Situ Lactonization in One Pot

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Benzotriazole as an Efficient Ligand in Cu-Catalyzed Glaser Reaction

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Regioselective radical arylation: silver-mediated synthesis of 3-phosphorylated coumarins, quinolin-2(1H)-one and benzophosphole oxides

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Exploring biological efficacy of coumarin clubbed thiazolo[3,2-b][1,2,4]triazoles as efficient inhibitors of urease: A biochemical and in silico approach

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Synthesis of Naphthols by Rh(III)-Catalyzed Domino C-H Activation, Annulation, and Lactonization Using Sulfoxonium Ylide as a Traceless Directing Group

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Copper-Catalyzed Three-Component Cascade Michael Addition/Heck-Type Alkylation/Annulation: Accessing Fully Substituted 1,3-Dihydro-2H-pyrrol-2-ones

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Developing new hybrid scaffold for urease inhibition based on carbazole-chalcone conjugates: Synthesis, assessment of therapeutic potential and computational docking analysis

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Copper-Catalyzed Cascade Cyclization Reaction of Enamines and Electron-Deficient Terminal Alkynes: Synthesis of Polysubstituted Pyrido[1,2-a]indoles

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Robust therapeutic potential of carbazole-triazine hybrids as a new class of urease inhibitors: A distinctive combination of nitrogen-containing heterocycles

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

Recent advances in synthesis and medicinal chemistry of benzodiazepines

1 reference

https://pubmed.ncbi.nlm.nih.gov/33398642

12 December 2020

10.1016/S0040-4039(00)91094-3

Identifiers

DOI

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:33398642%20AND%20SRC:MED&resulttype=core&format=json

9 January 2021

1 reference