(Q42732843)

6 November 2017

GSK6853, a Chemical Probe for Inhibition of the BRPF1 Bromodomain (English)

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6 November 2017

3

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6 November 2017

David J Fallon

9

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Chun-Wa Chung

5

object named as

Chun-Wa Chung

1 reference

6 November 2017

Paul Bamborough

1

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6 November 2017

Heather A Barnett

2

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6 November 2017

Mark J Bird

4

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6 November 2017

Peter D Craggs

6

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6 November 2017

Emmanuel H Demont

7

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6 November 2017

Hawa Diallo

8

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6 November 2017

Laurie J Gordon

10

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6 November 2017

Paola Grandi

11

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6 November 2017

Clare I Hobbs

12

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6 November 2017

Edward Hooper-Greenhill

13

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6 November 2017

Emma J Jones

14

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6 November 2017

Robert P Law

15

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6 November 2017

Armelle Le Gall

16

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6 November 2017

David Lugo

17

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6 November 2017

Anne-Marie Michon

18

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6 November 2017

Darren J Mitchell

19

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6 November 2017

Rab K Prinjha

20

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6 November 2017

Robert J Sheppard

21

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6 November 2017

Allan J B Watson

22

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6 November 2017

Robert J Watson

23

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6 November 2017

9 May 2016

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ACS Medicinal Chemistry Letters

6 November 2017

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6 November 2017

7

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6 November 2017

6

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6 November 2017

552-557

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Structure-Guided Design of IACS-9571, a Selective High-Affinity Dual TRIM24-BRPF1 Bromodomain Inhibitor

6 November 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4904261

Discovery of a Chemical Tool Inhibitor Targeting the Bromodomains of TRIM24 and BRPF.

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4904261

1,3-Dimethyl Benzimidazolones Are Potent, Selective Inhibitors of the BRPF1 Bromodomain

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4904261

Targeting bromodomains: epigenetic readers of lysine acetylation

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4904261

The MOZ histone acetyltransferase in epigenetic signaling and disease.

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4904261

Molecular insights into the recognition of N-terminal histone modifications by the BRPF1 bromodomain.

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4904261

BET bromodomain inhibitors: a patent review

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4904261

Discovery of epigenetic regulator I-BET762: lead optimization to afford a clinical candidate inhibitor of the BET bromodomains

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4904261

TET2 and TET3 regulate GlcNAcylation and H3K4 methylation through OGT and SET1/COMPASS

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4904261

Histone recognition and large-scale structural analysis of the human bromodomain family

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4904261

Recognition of unmodified histone H3 by the first PHD finger of bromodomain-PHD finger protein 2 provides insights into the regulation of histone acetyltransferases monocytic leukemic zinc-finger protein (MOZ) and MOZ-related factor (MORF)

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4904261

Getting physical in drug discovery II: the impact of chromatographic hydrophobicity measurements and aromaticity

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4904261

Discovery and characterization of small molecule inhibitors of the BET family bromodomains

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4904261

Suppression of inflammation by a synthetic histone mimic

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4904261

Selective inhibition of BET bromodomains

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4904261

Molecular basis of histone H3K36me3 recognition by the PWWP domain of Brpf1

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4904261

Molecular architecture of quartet MOZ/MORF histone acetyltransferase complexes

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4904261

The multidomain protein Brpf1 binds histones and is required for Hox gene expression and segmental identity

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4904261

Ligand efficiency: a useful metric for lead selection

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4904261

The maximal affinity of ligands

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4904261

A computational procedure for determining energetically favorable binding sites on biologically important macromolecules

27 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4904261

10.1021/ACSMEDCHEMLETT.6B00092

27 May 2018

Identifiers

DOI

1 reference

6 November 2017

1 reference

6 November 2017

PubMed publication ID

27326325

1 reference