(Q35285730)

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20 February 2020

title

Cell-based protein stabilization assays for the detection of interactions between small-molecule inhibitors and BRD4 (English)

1 reference

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Amaury E Fernández-Montalván

20 February 2020

author

4

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20 February 2020

Ben Bader

8

1 reference

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20 February 2020

author name string

Jessica Schulze

1

1 reference

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20 February 2020

Dieter Moosmayer

2

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20 February 2020

Joerg Weiske

3

1 reference

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20 February 2020

Christopher Herbst

5

1 reference

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20 February 2020

Marie Jung

6

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20 February 2020

Bernard Haendler

7

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20 February 2020

publication date

29 September 2014

1 reference

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Journal of Biomolecular Screening

20 February 2020

published in

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20 February 2020

volume

20

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20 February 2020

issue

2

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20 February 2020

page(s)

180-189

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Intracellular protein degradation in mammalian and bacterial cells

20 February 2020

cites work

1 reference

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High-density miniaturized thermal shift assays as a general strategy for drug discovery

21 January 2018

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Monitoring drug target engagement in cells and tissues using the cellular thermal shift assay.

21 January 2018

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Pulse proteolysis: A simple method for quantitative determination of protein stability and ligand binding

21 January 2018

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Identification of Direct Protein Targets of Small Molecules

21 January 2018

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Simplified proteomics approach to discover protein-ligand interactions.

21 January 2018

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Beta galactosidase complementation: a cell-based luminescent assay platform for drug discovery

21 January 2018

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HTRF: A technology tailored for drug discovery - a review of theoretical aspects and recent applications

21 January 2018

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Histone recognition and large-scale structural analysis of the human bromodomain family

21 January 2018

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Bromodomains and their pharmacological inhibitors

21 January 2018

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Targeting bromodomains: epigenetic readers of lysine acetylation

21 January 2018

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Affinity map of bromodomain protein 4 (BRD4) interactions with the histone H4 tail and the small molecule inhibitor JQ1.

21 January 2018

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A Simple Statistical Parameter for Use in Evaluation and Validation of High Throughput Screening Assays

21 January 2018

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Inhibitors of the proteasome block the degradation of most cell proteins and the generation of peptides presented on MHC class I molecules

21 January 2018

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Application of high-throughput isothermal denaturation to assess protein stability and screen for ligands

21 January 2018

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Chemical screening methods to identify ligands that promote protein stability, protein crystallization, and structure determination

21 January 2018

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A one-day, dispense-only IP-One HTRF assay for high-throughput screening of Galphaq protein-coupled receptors: towards cells as reagents

21 January 2018

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Different orientations of low-molecular-weight fragments in the binding pocket of a BRD4 bromodomain

21 January 2018

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Regulation of mammalian autophagy in physiology and pathophysiology.

21 January 2018

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Inhibition of eukaryotic translation elongation by cycloheximide and lactimidomycin

21 January 2018

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A beta oligomers - a decade of discovery

21 January 2018

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A noncompetitive small molecule inhibitor of estrogen-regulated gene expression and breast cancer cell growth that enhances proteasome-dependent degradation of estrogen receptor {alpha}.

21 January 2018

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Identification and characterization of pharmacological chaperones to correct enzyme deficiencies in lysosomal storage disorders

21 January 2018

1 reference

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21 January 2018

Identifiers

DOI

10.1177/1087057114552398

1 reference

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20 February 2020

1 reference

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